SCHEMBL7130463

SCHEMBL7130463

N=C(N)NCCC[C@H](N)C(=O)N(C(=O)OCc1ccccc1)[C@@H](CCCNC(=N)N)C(=O)Nc1ccc2ccccc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 7/20 0.39
ANPEP P15144 1/20 0.38
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C19 P33261 2/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 1/20 0.37
ROCK2 O75116 2/20 0.36
EPHX1 P07099 2/20 0.36
DPP8 Q6V1X1 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
PTGER4 P35408 1/20 0.35
SLC1A3 P43003 1/20 0.35
SLC1A1 P43005 1/20 0.35
PLAU P00749 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10649078 0.86 ROCK2 (0.36) LTA4HCYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL5052608 0.85 KMT2A (0.41) LTA4HANPEPALDH1A1LMNAMAPT
SCHEMBL10689300 0.85 CYP1A2 (0.37) LTA4HCYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL4727444 0.83 RAB9A (0.45) ALDH1A1MAPTSMN1; SMN2HSD17B10
SCHEMBL27892485 0.82 NPY4R (0.42) LTA4HANPEPDPP8DPP7SLC1A3
SCHEMBL10948492 0.80 FNTA (0.34) LMNAMAPTSMN1; SMN2EPHX1DPP8
SCHEMBL29517152 0.80 FOLH1 (0.42) LTA4HANPEPDPP8DPP7SLC1A3
SCHEMBL8362644 0.80 EPHX1 (0.39) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL7859247 0.80 EPHX1 (0.39) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL8336616 0.80 PTGER4 (0.36) LTA4HCYP1A2CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1278552-A2 FUNCTIONAL MRI AGENTS FOR CANCER IMAGING RESEARCH CORPORATION TECHNOLOGIES (US) 2003-01-29 EP disclosed
WO-2002080757-A2 NOVEL FUNCTIONAL AGENTS FOR MAGNETIC RESONANCE IMAGING METAPROBE, INC. (US) 2002-10-17 WO disclosed
WO-2001082976-A2 FUNCTIONAL MRI AGENTS FOR CANCER IMAGING RESEARCH CORPORATION TECHNOLOGIES (US) 2001-11-08 WO disclosed