SCHEMBL7136362

SCHEMBL7136362

CO/C=C(/C(=O)OC)c1ccccc1/C=C/C=C/c1ccc(F)cc1F

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 4/20 0.44
AR P10275 1/20 0.40
HTR2A P28223 2/20 0.39
HTR2C P28335 2/20 0.39
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
RELA Q04206 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7136772 1.00 NFE2L2 (0.44) NFE2L2ARHTR2AHTR2CPOLB
SCHEMBL7135431 0.91 NFE2L2 (0.44) NFE2L2ARHTR2AHTR2CRELA
SCHEMBL7135430 0.91 NFE2L2 (0.44) NFE2L2ARHTR2AHTR2CRELA
SCHEMBL7140087 0.88 AR (0.39) ARMAPTRAB9ARELA
SCHEMBL7140095 0.88 AR (0.39) ARMAPTRAB9ARELA
SCHEMBL7142993 0.86 KDM4E (0.38) MAPTKCNH2
SCHEMBL7142991 0.86 KDM4E (0.38) MAPTKCNH2
SCHEMBL7135427 0.86 MAOB (0.43) NFE2L2ARMAPT
SCHEMBL7133655 0.86 MAOB (0.43) NFE2L2ARMAPT
SCHEMBL10358886 0.81 SNCA (0.45) NFE2L2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0996439-B1 BETA-ALKOXYACRYLATES AGAINST MALARIA HOFFMANN LA ROCHE (CH) 2003-01-08 EP claimed
EP-0996439-B1 BETA-ALKOXYACRYLATES AGAINST MALARIA HOFFMANN LA ROCHE (CH) 2003-01-08 EP disclosed
US-6084120-A ACTIVE AGAINST CHLOROQUINE-SENSITIVE PATIENTS AND AGAINST CHLOROQUINE-RESISTANT MALARIA PATHOGENS; PROPHYLAXIS AND TREATMENT; E.G., A 3 METHOXY-2-(2-(4-PHENYLBUTA-1,3-DIEN-1-YL)PHENYL)ACRYLIC ACID HOFFMANN-LA ROCHE INC. (US) 2000-07-04 US disclosed