SCHEMBL7140087

SCHEMBL7140087

CO/C=C(/C(=O)OC)c1ccccc1/C=C/C=C/c1ccc(F)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.39
NOS2 P35228 1/20 0.36
RELA Q04206 1/20 0.35
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ABCG2 Q9UNQ0 2/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7140095 1.00 AR (0.39) ARNOS2RELANPC1MAPT
SCHEMBL7164686 0.91 AR (0.39) ARNOS2RELAMAPTABCG2
SCHEMBL7164682 0.91 AR (0.39) ARNOS2RELAMAPTABCG2
SCHEMBL7136362 0.88 NFE2L2 (0.44) ARRELAMAPTRAB9A
SCHEMBL7133616 0.88 PTPN5 (0.44) NPC1MAPTHPGDRAB9ASMN1; SMN2
SCHEMBL7133619 0.88 PTPN5 (0.44) NPC1MAPTHPGDRAB9ASMN1; SMN2
SCHEMBL7136772 0.88 NFE2L2 (0.44) ARRELAMAPTRAB9A
SCHEMBL7140245 0.87 RAB9A (0.39) RELANPC1MAPTHPGDRAB9A
SCHEMBL7140250 0.87 RAB9A (0.39) RELANPC1MAPTHPGDRAB9A
SCHEMBL7135427 0.84 MAOB (0.43) ARMAPTSMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0996439-B1 BETA-ALKOXYACRYLATES AGAINST MALARIA HOFFMANN LA ROCHE (CH) 2003-01-08 EP claimed
US-6084120-A ACTIVE AGAINST CHLOROQUINE-SENSITIVE PATIENTS AND AGAINST CHLOROQUINE-RESISTANT MALARIA PATHOGENS; PROPHYLAXIS AND TREATMENT; E.G., A 3 METHOXY-2-(2-(4-PHENYLBUTA-1,3-DIEN-1-YL)PHENYL)ACRYLIC ACID HOFFMANN-LA ROCHE INC. (US) 2000-07-04 US claimed
EP-0996439-B1 BETA-ALKOXYACRYLATES AGAINST MALARIA HOFFMANN LA ROCHE (CH) 2003-01-08 EP disclosed
US-6084120-A ACTIVE AGAINST CHLOROQUINE-SENSITIVE PATIENTS AND AGAINST CHLOROQUINE-RESISTANT MALARIA PATHOGENS; PROPHYLAXIS AND TREATMENT; E.G., A 3 METHOXY-2-(2-(4-PHENYLBUTA-1,3-DIEN-1-YL)PHENYL)ACRYLIC ACID HOFFMANN-LA ROCHE INC. (US) 2000-07-04 US disclosed