SCHEMBL7137103

SCHEMBL7137103

CN(C)CCc1cccc(-c2nc3cccc(C(N)=O)c3[nH]2)c1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.55
PIM1 P11309 2/20 0.48
PIM3 Q86V86 2/20 0.48
AURKB Q96GD4 2/20 0.48
DYRK3 O43781 1/20 0.48
MAP4K4 O95819 1/20 0.48
RPS6KB1 P23443 1/20 0.48
CSNK2A1 P68400 1/20 0.48
PKN2 Q16513 1/20 0.48
BRSK1 Q8TDC3 1/20 0.48
HIPK2 Q9H2X6 1/20 0.48
CLK4 Q9HAZ1 1/20 0.48
MKNK2 Q9HBH9 1/20 0.48
STK17A Q9UEE5 1/20 0.48
MAP4K5 Q9Y4K4 1/20 0.48
CHEK2 O96017 1/20 0.45
HTR7 P34969 2/20 0.44
DNMT3B Q9UBC3 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7140624 0.89 PARP1 (0.48) PARP1PIM1PIM3AURKBDYRK3
SCHEMBL7131933 0.89 PARP1 (0.54) PARP1PIM1PIM3AURKBDYRK3
SCHEMBL7136552 0.86 PARP1 (0.52) PARP1PIM1PIM3AURKB
SCHEMBL7141044 0.85 PARP1 (0.48) PARP1PIM1PIM3AURKB
SCHEMBL7137094 0.83 PARP1 (0.80) PARP1PIM1PIM3AURKBDYRK3
SCHEMBL3577822 0.82 MAP4K4 (0.72) PARP1PIM1PIM3AURKBDYRK3
SCHEMBL7139317 0.81 PARP1 (0.58) PARP1PIM1PIM3AURKBBRSK1
SCHEMBL6379938 0.80 PKN2 (0.41) PARP1PIM1PIM3AURKBDYRK3
SCHEMBL7132446 0.80 PARP1 (0.59) PARP1PIM1PIM3AURKBBRSK1
SCHEMBL29696369 0.79 NPC1 (0.53) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6509365-B1 2-phenylbenzimidazoles and 2-phenylindoles, and production and use thereof BASF AKTIENGESELLSCHAFT (DE) 2003-01-21 US disclosed