SCHEMBL7141044

SCHEMBL7141044

CNCCc1cccc(-c2nc3cccc(C(N)=O)c3[nH]2)c1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 17/20 0.48
PIM1 P11309 1/20 0.43
PIM3 Q86V86 1/20 0.43
AURKB Q96GD4 1/20 0.43
MMP2 P08253 2/20 0.41
MMP9 P14780 2/20 0.41
MMP8 P22894 2/20 0.41
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7136552 0.86 PARP1 (0.52) PARP1PIM1PIM3AURKBMMP2
SCHEMBL7137103 0.85 PARP1 (0.55) PARP1PIM1PIM3AURKB
SCHEMBL7140624 0.83 PARP1 (0.48) PARP1PIM1PIM3AURKB
SCHEMBL7141034 0.83 PARP1 (0.72) PARP1
SCHEMBL7139317 0.81 PARP1 (0.58) PARP1PIM1PIM3AURKB
SCHEMBL7132446 0.80 PARP1 (0.59) PARP1PIM1PIM3AURKB
SCHEMBL29696369 0.79 NPC1 (0.53) PARP1CYP3A4CYP2C9
SCHEMBL7137491 0.78 PARP1 (0.47) PARP1
SCHEMBL3585144 0.78 PARP1 (0.64) PARP1PIM1AURKB
SCHEMBL3579908 0.77 PARP1 (0.61) PARP1PIM1PIM3AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6509365-B1 2-phenylbenzimidazoles and 2-phenylindoles, and production and use thereof BASF AKTIENGESELLSCHAFT (DE) 2003-01-21 US disclosed