SCHEMBL7137997

SCHEMBL7137997

CSc1ccc(C=C2C(=O)Nc3c(Br)cc(Br)c(C)c32)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.44
ALDH1A1 P00352 3/20 0.37
POLB P06746 1/20 0.37
RET P07949 1/20 0.36
MAPT P10636 4/20 0.35
GAA P10253 1/20 0.34
SIRT1 Q96EB6 2/20 0.34
SIRT2 Q8IXJ6 1/20 0.34
SIRT3 Q9NTG7 1/20 0.34
PSMB2 P49721 1/20 0.34
EGFR P00533 1/20 0.34
CYP1A2 P05177 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
DRD1 P21728 1/20 0.34
PTGS1 P23219 1/20 0.34
MAPK1 P28482 1/20 0.34
PTGS2 P35354 1/20 0.34
OPRM1 P35372 1/20 0.34
PPARG P37231 1/20 0.34
PSEN1 P49768 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7138182 0.87 KMT2A (0.42) ALDH1A1RETMAPTSIRT1SIRT2
SCHEMBL7138862 0.87 MAPT (0.47) ALDH1A1POLBRETMAPTSIRT1
SCHEMBL7135160 0.85 METAP1 (0.50) ALDH1A1POLBRETMAPTSIRT2
SCHEMBL7136076 0.85 LRRK2 (0.42) GSK3BSIRT1SIRT2SIRT3PSEN1
SCHEMBL7133993 0.85 METAP1 (0.50) GSK3BALDH1A1POLBRETMAPT
SCHEMBL7136101 0.84 RET (0.44) POLBRETGAASIRT1SIRT2
SCHEMBL7131272 0.82 SIRT2 (0.52) ALDH1A1POLBRETMAPTSIRT1
SCHEMBL7138840 0.82 RET (0.55) ALDH1A1RETMAPTGAASIRT1
SCHEMBL7138260 0.82 METAP1 (0.55) GSK3BPOLBRETMETAP1
SCHEMBL7138851 0.82 IGF1R (0.44) ALDH1A1RETMAPTGAASIRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6506763-B2 Useful in prevention and treatment of protein kinase related disorders such as cancer SUGEN, INC. 2003-01-14 US disclosed