SCHEMBL7140412

SCHEMBL7140412

CCCCCNCc1cccc(-c2ccc(-c3ccccc3)[nH]2)c1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.55
CYP2D6 P10635 3/20 0.55
CYP2C19 P33261 3/20 0.55
HRH4 Q9H3N8 1/20 0.49
HRH3 Q9Y5N1 1/20 0.49
SIGMAR1 Q99720 4/20 0.48
MAOA P21397 1/20 0.46
CHRM2 P08172 3/20 0.45
SMN1; SMN2 Q16637 1/20 0.43
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
VSIR Q9H7M9 1/20 0.42
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29864521 0.84 CYP1A2 (0.64) CYP1A2CYP2D6CYP2C19HRH4HRH3
SCHEMBL7140600 0.83 SCN2A (0.52) CYP1A2CYP2D6CYP2C19HRH4HRH3
SCHEMBL7143456 0.82 SCN2A (0.51) CYP1A2CYP2D6CYP2C19HRH4HRH3
SCHEMBL8189931 0.79 SCN2A (0.50) CYP1A2CYP2D6CYP2C19CNR1CNR2
SCHEMBL21648321 0.78 CYP1A2 (0.59) CYP1A2CYP2D6CYP2C19HRH4HRH3
SCHEMBL9257479 0.77 CYP1A2 (0.76) CYP1A2CYP2D6CYP2C19HRH4HRH3
SCHEMBL15859362 0.77 CYP1A2 (0.76) CYP1A2CYP2D6CYP2C19HRH4HRH3
SCHEMBL538475 0.77 MAOA (0.76) CYP1A2CYP2D6CYP2C19HRH4HRH3
Hydrochloric Acid SCHEMBL29692481 0.77 CYP1A2 (0.62) CYP1A2CYP2D6CYP2C19HRH4HRH3
SCHEMBL16436983 0.76 CYP1A2 (0.61) CYP1A2CYP2D6CYP2C19HRH4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6515133-B1 Certain diaryl imidazoles act as partial agonists or antagonists for NPY receptors, in particular NPY 5 receptors. They are of use, for example in treating loss of appetite. Such compounds bear aryl groups in the 2 position. NEUROGEN CORPORATION 2003-02-04 US disclosed