SCHEMBL7140882

SCHEMBL7140882

CCCC(C(=O)O)N(CCOC)CCOC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.43
AKR1A1 P14550 1/20 0.43
CHRM3 P20309 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
ADRA1A P35348 1/20 0.43
HRH1 P35367 1/20 0.43
DRD3 P35462 1/20 0.43
SLC6A3 Q01959 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
GABRA1 P14867 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GRIK1 P39086 1/20 0.39
SLC1A3 P43003 1/20 0.39
SLC1A2 P43004 1/20 0.39
SLC1A1 P43005 1/20 0.39
GRIK2 Q13002 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7144010 1.00 CHRM1 (0.43) CHRM1AKR1A1CHRM3HTR2AHTR2C
Hydrochloric Acid SCHEMBL7431962 0.98 CHRM1 (0.42) CHRM1AKR1A1CHRM3HTR2AHTR2C
SCHEMBL7140120 0.89 CA2 (0.40) GABRA1GABRG2GABRB3GRIK1SLC1A3
SCHEMBL5718295 0.89 GABRA1 (0.39) GABRA1GABRG2GABRB3NOD1PIK3CD
SCHEMBL7136332 0.85 GABRA1 (0.49) GABRA1GABRG2GABRB3PIK3CDALDH1A1
SCHEMBL7140859 0.85 GABRA1 (0.49) GABRA1GABRG2GABRB3PIK3CDALDH1A1
SCHEMBL5718181 0.84 GABRA1 (0.38) GABRA1GABRG2GABRB3NOD1TSHR
SCHEMBL5718288 0.82 GABRA1 (0.40) GABRA1GABRG2GABRB3PIK3CDALDH1A1
SCHEMBL3783724 0.82 CHRM1 (0.52) CHRM1AKR1A1CHRM3HTR2AHTR2C
SCHEMBL12932066 0.82 CHRM1 (0.52) CHRM1AKR1A1CHRM3HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1098871-B1 alpha-AMINO ACID PHENYL ESTER DERIVATIVES AKZO NOBEL NV (NL) 2003-07-09 EP disclosed
US-6451854-B1 α-amino acid phenyl ester derivatives AKZO NOBEL N.V. (NL) 2002-09-17 US disclosed
EP-1098871-A1 $g(a)-AMINO ACID PHENYL ESTER DERIVATIVES Akzo Nobel N.V. (NL) 2001-05-16 EP disclosed
WO-2000005196-A1 α-AMINO ACID PHENYL ESTER DERIVATIVES AKZO NOBEL N.V. (NL) 2000-02-03 WO disclosed