SCHEMBL7141409

SCHEMBL7141409

CCOc1ccc([S+]([O-])N2CCN(CC)CC2)cc1C#N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 1/20 0.37
KCNH2 Q12809 1/20 0.37
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
KDM4E B2RXH2 2/20 0.35
NPY2R P49146 1/20 0.35
ALDH1A1 P00352 5/20 0.34
XDH P47989 1/20 0.34
AR P10275 2/20 0.33
MTOR P42345 1/20 0.33
HPGD P15428 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
PRMT5 O14744 1/20 0.31
WDR77 Q9BQA1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7006925 0.89 KCNJ1 (0.37) KCNJ1KCNH2NOS3NOS1NOS2
SCHEMBL12380552 0.76 NPC1 (0.49) KCNJ1KCNH2KDM4EALDH1A1MAPT
SCHEMBL1231574 0.74 TSHR (0.57) ALDH1A1MAPTSMN1; SMN2KMT2A
SCHEMBL12380568 0.68 CHKA (0.56) KCNJ1KCNH2KDM4EALDH1A1HPGD
SCHEMBL456337 0.67 ALDH1A1 (0.44) ALDH1A1XDHSMN1; SMN2MEN1KMT2A
SCHEMBL7003806 0.67 KMT2A (0.41) ALDH1A1MAPTSMN1; SMN2MEN1KMT2A
SCHEMBL13181116 0.67 GAA (0.53) NOS3NOS1NOS2KDM4EALDH1A1
SCHEMBL7003402 0.66 MAPK1 (0.41) KCNH2MAPTSMN1; SMN2MEN1KMT2A
SCHEMBL4694901 0.65 AR (0.57) KDM4EALDH1A1XDHARHPGD
SCHEMBL1197763 0.64 MAPT (0.54) NOS2KDM4EALDH1A1XDHAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1292586-A1 PROCESS FOR THE PREPARATION OF PYRAZOLOPYRIMIDINONES Pfizer Limited (GB) 2003-03-19 EP disclosed
WO-2001098284-A1 PROCESS FOR THE PREPARATION OF PYRAZOLOPYRIMIDINONES PFIZER LIMITED (GB) 2001-12-27 WO disclosed