SCHEMBL7142236

SCHEMBL7142236

Nc1ccc(S(=O)(=O)c2cc(-c3cccc(C(F)(F)F)c3)nc(N3CCCC3)c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.56
HTR2A P28223 1/20 0.56
PIK3CA P42336 7/20 0.47
AKT1 P31749 1/20 0.47
MTOR P42345 1/20 0.47
HTR1D P28221 1/20 0.47
HTR2C P28335 1/20 0.47
PIK3C3 Q8NEB9 2/20 0.46
MEN1 O00255 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 1/20 0.46
THRB P10828 2/20 0.44
LMNA P02545 2/20 0.44
MAPT P10636 1/20 0.43
XDH P47989 1/20 0.43
CNR2 P34972 1/20 0.43
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
ATM Q13315 1/20 0.42
AR P10275 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7143107 0.90 HTR6 (0.59) HTR6HTR2APIK3CAAKT1MTOR
SCHEMBL7138600 0.84 HTR6 (0.65) HTR6HTR2APIK3CAAKT1MTOR
SCHEMBL7140803 0.84 HTR6 (0.59) HTR6HTR2APIK3CAAKT1MTOR
SCHEMBL7143113 0.81 HTR6 (0.56) HTR6HTR2APIK3CAAKT1MTOR
SCHEMBL7137463 0.81 HTR6 (0.56) HTR6HTR2APIK3CAAKT1MTOR
SCHEMBL7143666 0.81 HTR6 (0.60) HTR6HTR2APIK3CAAKT1MTOR
SCHEMBL7143714 0.80 HTR6 (0.62) HTR6HTR2APIK3CAAKT1MTOR
SCHEMBL7140658 0.78 HTR6 (0.62) HTR6HTR2APIK3CAAKT1MTOR
SCHEMBL7140758 0.78 HTR6 (0.62) HTR6HTR2APIK3CAAKT1MTOR
SCHEMBL7136657 0.77 HTR6 (0.61) HTR6HTR2APIK3CAAKT1MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0930302-B1 Benzosulfone derivatives HOFFMANN LA ROCHE (CH) 2003-04-02 EP disclosed
US-5990105-A POSSESS A SELECTIVE AFFINITY TO 5HT-6 RECEPTORS; TREATING OR PREVENTING PSYCHOSES, SCHIZOPHRENIA, MANIC DEPRESSIONS, DEPRESSIONS, NEUROLOGICAL DISORDERS, PARKINSON'S, AMYOTROPHIC LATERAL SCLEROSIS, ALZHEIMER'S AND HUNTINGTON'S DISEASE HOFFMANN-LA ROCHE INC. (US) 1999-11-23 US disclosed
EP-0930302-A2 Benzosulfone derivatives F.HOFFMANN-LA ROCHE AG (CH) 1999-07-21 EP disclosed