SCHEMBL7144713

SCHEMBL7144713

O=C(c1ccc(Cl)cc1)C(Br)c1cccnc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.53
CYP11B1 P15538 1/20 0.49
CYP11B2 P19099 1/20 0.49
KMT2A Q03164 5/20 0.48
ALOX15 P16050 1/20 0.48
NAMPT P43490 1/20 0.47
CYP3A4 P08684 1/20 0.45
CYP3A5 P20815 1/20 0.45
MEN1 O00255 3/20 0.45
ALDH1A1 P00352 2/20 0.45
LMNA P02545 2/20 0.45
USP2 O75604 1/20 0.45
MAPT P10636 2/20 0.43
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
TSHR P16473 1/20 0.43
SUCNR1 Q9BXA5 2/20 0.42
FFAR2 O15552 1/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL6284312 0.98 CYP19A1 (0.51) CYP19A1CYP11B1CYP11B2KMT2AALOX15
SCHEMBL7149156 0.86 CYP17A1 (0.49) CYP19A1KMT2AALDH1A1LMNAMAPT
SCHEMBL7140967 0.86 SMN1; SMN2 (0.51) NAMPTALDH1A1LMNASMN1; SMN2GAA
SCHEMBL7149214 0.85 POLB (0.51) CYP11B1CYP11B2KMT2AMEN1ALDH1A1
SCHEMBL7142799 0.85 NAMPT (0.49) KMT2ANAMPTALDH1A1LMNAMAPT
Bromide SCHEMBL6279795 0.85 CYP17A1 (0.48) CYP19A1KMT2AALDH1A1LMNAMAPT
Bromide SCHEMBL6282444 0.84 SMN1; SMN2 (0.50) NAMPTALDH1A1LMNASMN1; SMN2GAA
SCHEMBL7141524 0.84 NPSR1 (0.52) KMT2AALOX15CYP3A4MEN1ALDH1A1
Bromide SCHEMBL6283209 0.84 POLB (0.50) CYP11B1CYP11B2KMT2AMEN1ALDH1A1
Bromide SCHEMBL6276160 0.84 NAMPT (0.48) KMT2ANAMPTALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6620825-B1 1,3-Azole compound substituted by pyridyl; administering as antiasthmatic, antiinflammatory or antiallergen agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-16 US disclosed
US-6436966-B1 Adenosine A3 receptor antagonists TAKEDA CHEMICAL IND., LTD. (JP) 2002-08-20 US disclosed