SCHEMBL7140967

SCHEMBL7140967

O=C(c1ccccc1)C(Br)c1cccnc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.51
ALDH1A1 P00352 2/20 0.50
APP P05067 1/20 0.50
GAA P10253 1/20 0.50
HCAR3 P49019 1/20 0.50
HCAR2 Q8TDS4 1/20 0.50
CFTR P13569 1/20 0.50
SLC6A2 P23975 1/20 0.50
SLC6A4 P31645 1/20 0.50
SLC6A3 Q01959 1/20 0.50
GOPC Q9HD26 1/20 0.50
HTT P42858 1/20 0.49
EPHX2 P34913 2/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
PLOD2 O00469 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
LMNA P02545 2/20 0.46
CES2 O00748 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL6282444 0.98 SMN1; SMN2 (0.50) SMN1; SMN2ALDH1A1APPGAAHCAR3
SCHEMBL7147666 0.90 ALDH1A1 (0.55) SMN1; SMN2ALDH1A1APPGAAHCAR3
Bromide SCHEMBL6546257 0.89 ALDH1A1 (0.53) SMN1; SMN2ALDH1A1APPGAAHCAR3
SCHEMBL7149156 0.87 CYP17A1 (0.49) SMN1; SMN2ALDH1A1APPGAAHCAR3
SCHEMBL7142799 0.86 NAMPT (0.49) SMN1; SMN2ALDH1A1GAALMNATBXAS1
SCHEMBL7149214 0.86 POLB (0.51) SMN1; SMN2ALDH1A1GAAEPHX2LMNA
Bromide SCHEMBL6279795 0.86 CYP17A1 (0.48) SMN1; SMN2ALDH1A1APPGAAHCAR3
SCHEMBL7144713 0.86 CYP19A1 (0.53) SMN1; SMN2ALDH1A1GAAHTTL3MBTL1
Bromide SCHEMBL6284312 0.84 CYP19A1 (0.51) SMN1; SMN2ALDH1A1GAAHTTL3MBTL1
Bromide SCHEMBL6283209 0.84 POLB (0.50) SMN1; SMN2ALDH1A1GAAEPHX2KCNA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6620825-B1 1,3-Azole compound substituted by pyridyl; administering as antiasthmatic, antiinflammatory or antiallergen agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-16 US disclosed
US-6436966-B1 Adenosine A3 receptor antagonists TAKEDA CHEMICAL IND., LTD. (JP) 2002-08-20 US disclosed
EP-0149884-B1 5-PYRIDYL-1,3-THIAZOLE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1992-12-16 EP disclosed
US-4612321-A 5-pyridyl-1,3-thiazole derivatives TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 1986-09-16 US disclosed
EP-0149884-A2 5-Pyridyl-1,3-thiazole derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1985-07-31 EP disclosed
US-3940486-A Imidazole derivatives in the treatment of pain CIBA-GEIGY CORPORATION (US) 1976-02-24 US disclosed