SCHEMBL7144794

SCHEMBL7144794

CS(=O)(=O)N1CC(S)CC1CCOc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 1/20 0.41
HCRTR1 O43613 1/20 0.37
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
KDM4E B2RXH2 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TEAD1 P28347 1/20 0.36
TEAD3 Q99594 1/20 0.36
TAAR1 Q96RJ0 1/20 0.35
HTR1A P08908 1/20 0.35
HTR7 P34969 1/20 0.35
MMP8 P22894 1/20 0.35
MMP13 P45452 1/20 0.35
ADAM17 P78536 1/20 0.35
KCNA3 P22001 1/20 0.35
PLA2G7 Q13093 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5415653 1.00 ECE1 (0.41) ECE1HCRTR1ALDH1A1MEN1HTT
SCHEMBL5407509 0.86 ECE1 (0.42) ECE1MMP8MMP13
SCHEMBL7137605 0.86 ECE1 (0.42) ECE1MMP8MMP13
SCHEMBL5405292 0.74 DRD2 (0.43) ECE1MEN1KMT2A
SCHEMBL5399402 0.73 ECE1 (0.45) ECE1ALDH1A1HTTKMT2ASMN1; SMN2
Trifluoroacetic Acid SCHEMBL5404968 0.72 ECE1 (0.36) ECE1KDM4E
SCHEMBL7148484 0.72 NPC1 (0.49) HCRTR1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL7140645 0.70 ECE1 (0.33) ECE1
SCHEMBL5411627 0.70 ECE1 (0.43) ECE1
SCHEMBL5406301 0.69 KMT2A (0.36) ECE1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303486-A1 PYRROLIDINE DERIVATIVES AS METALLOPROTEASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2003-04-23 EP disclosed
WO-2002008185-A1 PYRROLIDINE DERIVATIVES AS METALLOPROTEASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2002-01-31 WO disclosed