SCHEMBL7145669

SCHEMBL7145669

COc1cc2c(cc1OC)CC(NCC(N)=O)C2

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 3/20 0.41
ADRB2 P07550 1/20 0.41
CYP2C9 P11712 2/20 0.40
CYP2D6 P10635 1/20 0.40
ALOX15 P16050 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39
KDM4E B2RXH2 1/20 0.38
PDE4B Q07343 1/20 0.38
NQO2 P16083 1/20 0.37
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11005852 0.86 CA1 (0.50) CA1CA2KMT2AMEN1ALDH1A1
SCHEMBL11003933 0.81 ALDH1A1 (0.47) CA1CA2KMT2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL11003886 0.80 ALDH1A1 (0.46) CA1CA2KMT2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL7140757 0.78 KDM1A (0.36) CA1CA2ALDH1A1
SCHEMBL14198135 0.76 CA1 (0.53) CA1CA2KMT2AMEN1ALDH1A1
SCHEMBL27490005 0.76 CA1 (0.58) CA1CA2KMT2AMEN1KDM4E
SCHEMBL399565 0.75 KDM1A (0.50) CA1CA2ALDH1A1MTNR1AMTNR1B
Hydrochloric Acid SCHEMBL4869944 0.73 KDM1A (0.49) CA1CA2ALDH1A1MTNR1AMTNR1B
SCHEMBL8688541 0.73 DRD2 (0.56) CA1CA2ALDH1A1CYP2C9CYP2D6
SCHEMBL11896157 0.73 CA1 (0.54) CA1CA2KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0951465-B1 ALPHA-AMINO ACID AMIDES, PREPARATION THEREOF AND THE THERAPEUTICAL USE THEREOF CHIESI FARMA SPA (IT) 2003-04-16 EP disclosed
US-6114391-A A DERIVATIVES OF SERINAMIDE, GLYCINAMIDE, ALANINAMIDE AND PHENYLALANINAMIDE FOR TREATING NEUROLOGICAL DISEASES CHIESI FARMACEUTICI S.P.A. (IT) 2000-09-05 US disclosed