SCHEMBL7146905

SCHEMBL7146905

COC(=O)c1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1C

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.57
LMNA P02545 2/20 0.57
MAPT P10636 1/20 0.57
POLB P06746 2/20 0.53
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
PKM P14618 3/20 0.52
BRD4 O60885 1/20 0.52
KDM4E B2RXH2 3/20 0.52
HSD17B10 Q99714 2/20 0.52
HPGD P15428 1/20 0.52
CASP1 P29466 1/20 0.52
CASP7 P55210 1/20 0.52
HSD17B3 P37058 1/20 0.51
HSD17B2 P37059 1/20 0.51
TCF4 P15884 1/20 0.51
CTNNB1 P35222 1/20 0.51
GAA P10253 3/20 0.50
GLA P06280 1/20 0.50
ERAP1 Q9NZ08 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6979802 0.86 LMNA (0.60) ALDH1A1LMNAMAPTPOLBMEN1
SCHEMBL6979537 0.86 HSD17B3 (0.64) ALDH1A1LMNAMAPTPOLBMEN1
SCHEMBL6977966 0.82 MAPT (0.70) ALDH1A1LMNAMAPTPOLBMEN1
SCHEMBL15772389 0.82 MAPT (0.70) ALDH1A1LMNAMAPTPOLBMEN1
SCHEMBL6976969 0.81 LMNA (0.57) ALDH1A1LMNAMAPTPOLBMEN1
SCHEMBL16470144 0.80 ALDH1A1 (0.53) ALDH1A1LMNAMAPTPOLBKDM4E
SCHEMBL5101148 0.79 FFAR4 (0.69) ALDH1A1LMNAMAPTKDM4EHSD17B10
SCHEMBL5324234 0.79 KDM4E (0.59) ALDH1A1LMNAMAPTPOLBKDM4E
SCHEMBL25073129 0.78 PTPN11 (0.42) ALDH1A1LMNAMAPTPOLBMEN1
SCHEMBL25073301 0.78 RXFP1 (0.44) ALDH1A1LMNAMAPTPOLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6525050-B1 Inhibit the enzyme aminoimidazole carboxamide ribonucleotide formyl transferase; antiproliferative agents; antitumor, antiinflammatory, antipsoriatic, and/or immunosuppressive AGOURON PHARMACEUTICALS, INC. 2003-02-25 US disclosed