Triaziquone

Triaziquone

SCHEMBL7147458

CC1(C)CC(O)CC(C)(C)N1O.O=C(O)CC(O)(CC(=O)O)C(=O)O.O=C1C=C(N2CC2)C(=O)C(N2CC2)=C1N1CC1

nearest known ligand 0.31

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACVR1ADORA1ADORA2AADORA2BADORA3ESR1ESR2FLT3GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSC1HRH1HTR7IDH1IDH2IRAK1JAK1JAK2JAK3MEN1OPRM1P2RX3PDE5ASCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASIGMAR1SLC6A2SYKTACR1TOP2ATYK2

The experimentally established mechanism targets of Triaziquone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 2/20 0.31
SLC13A5 Q86YT5 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Triaziquone SCHEMBL2236656 0.85 ALDH1A1 (0.43) ALDH1A1KDM4ESLC13A5LMNAMAPT
Triaziquone SCHEMBL14237202 0.85 TP53 (0.35) ALDH1A1MAPT
Triaziquone SCHEMBL759304 0.82
Citric Acid SCHEMBL985329 0.80 ALDH1A1 (0.48) ALDH1A1KDM4ESLC13A5LMNAMAPT
Citric Acid SCHEMBL986854 0.80 ALDH1A1 (0.48) ALDH1A1KDM4ESLC13A5LMNAMAPT
Citric Acid SCHEMBL986838 0.80 ALDH1A1 (0.48) ALDH1A1KDM4ESLC13A5LMNAMAPT
Triaziquone SCHEMBL6236164 0.80 ALDH1A1 (0.36) ALDH1A1KDM4ESLC13A5LMNAMAPT
Edetic Acid SCHEMBL23361308 0.77 ALDH1A1 (0.35) ALDH1A1KDM4ESLC13A5LMNAMAPT
Triaziquone SCHEMBL5307413 0.77
Triaziquone SCHEMBL22346328 0.72 DNMT1 (0.39) LMNAMAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362083-A1 INK-JET INK AND RECORDING MATERIAL Ciba SC Holding AG (CH) 2003-11-19 EP disclosed
WO-2002055618-A1 INK-JET INK AND RECORDING MATERIAL CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2002-07-18 WO disclosed