SCHEMBL714749

SCHEMBL714749

Cc1c(F)ccc2cc(C(C)NC(=O)O)c(N3CCN(CC(F)(F)F)CC3)nc12

nearest known ligand 0.39

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 9/20 0.39
GPR6 P46095 10/20 0.35
SCN10A Q9Y5Y9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL715924 0.86 OPRK1 (0.41) OPRK1GPR6
SCHEMBL14481792 0.84 OPRK1 (0.39) OPRK1
SCHEMBL15875794 0.84 OPRK1 (0.40) OPRK1SCN10A
SCHEMBL14480924 0.84 OPRK1 (0.39) OPRK1GPR6
SCHEMBL14481349 0.84 MAPT (0.42) OPRK1
SCHEMBL717459 0.81 OPRK1 (0.38) OPRK1SCN10A
SCHEMBL15875802 0.81 OPRK1 (0.38) OPRK1SCN10A
SCHEMBL14481180 0.80 CHRNA7 (0.45)
SCHEMBL715385 0.80 OPRK1 (0.43) OPRK1GPR6
SCHEMBL11378 0.80 KDM4E (0.39) OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2403847-B1 TRIAZINE DERIVATIVES AS KINASE INHIBITORS UCB BIOPHARMA SPRL (BE) 2016-03-02 EP disclosed
US-8785628-B2 Triazine derivatives as kinase inhibitors UCB PHARMA, S.A. (BE) 2014-07-22 US disclosed
US-20120053167-A1 Triazine Derivatives as Kinase Inhibitors UCB PHARMA, S.A. (BE) 2012-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120053167-A1 Triazine Derivatives as Kinase Inhibitors MAP3K15, PI4KA, MAP3K20 OPRK1 416/4885GPR6 2471/4885SCN10A 2325/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.