SCHEMBL7148265

SCHEMBL7148265

Cc1cccc(C(=O)C(Br)c2cccnc2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.49
ELANE P08246 2/20 0.45
VNN1 O95497 1/20 0.44
CTSL P07711 1/20 0.44
CTSS P25774 1/20 0.44
LMNA P02545 1/20 0.44
BRAF P15056 1/20 0.44
IDE P14735 1/20 0.44
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
NT5E P21589 1/20 0.43
GRM5 P41594 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL6284648 0.99 NPC1 (0.50) NPC1RAB9AKMT2AMEN1ALDH1A1
SCHEMBL7142887 0.89 TDP1 (0.47) NPC1RAB9AKMT2AMEN1ALDH1A1
Bromide SCHEMBL6279797 0.87 TDP1 (0.46) NPC1RAB9AKMT2AMEN1ALDH1A1
SCHEMBL7142799 0.84 NAMPT (0.49) NPC1RAB9AKMT2AALDH1A1MAPT
SCHEMBL7143390 0.84 NT5E (0.52) NPC1RAB9AKMT2AALDH1A1ELANE
SCHEMBL17762880 0.84 PARP1 (0.50) NPC1RAB9AKMT2AMEN1TDP1
Hydrochloric Acid SCHEMBL11477585 0.83 NPC1 (0.48) NPC1RAB9AKMT2AMEN1ALDH1A1
SCHEMBL7141524 0.83 NPSR1 (0.52) NPC1RAB9AKMT2AMEN1ALDH1A1
Bromide SCHEMBL6283062 0.83 NT5E (0.51) NPC1RAB9AKMT2AALDH1A1ELANE
Bromide SCHEMBL6276160 0.83 NAMPT (0.48) NPC1RAB9AKMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6620825-B1 1,3-Azole compound substituted by pyridyl; administering as antiasthmatic, antiinflammatory or antiallergen agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-16 US disclosed
US-6436966-B1 Adenosine A3 receptor antagonists TAKEDA CHEMICAL IND., LTD. (JP) 2002-08-20 US disclosed