SCHEMBL7148745

SCHEMBL7148745

NN=Cc1ccc(CNC(=O)[C@@H]2CCCN2C(=O)[C@H](N)Cc2ccccc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
PKM P14618 1/20 0.52
CYP2C19 P33261 1/20 0.52
ALDH1A1 P00352 1/20 0.52
F2 P00734 4/20 0.52
DPP4 P27487 3/20 0.50
DPP8 Q6V1X1 2/20 0.50
DPP9 Q86TI2 2/20 0.50
DPP7 Q9UHL4 2/20 0.50
FAP Q12884 1/20 0.50
OPRM1 P35372 2/20 0.48
OPRD1 P41143 1/20 0.48
NPC1 O15118 1/20 0.48
POLB P06746 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27544517 1.00 CYP3A4 (0.52) CYP3A4CYP2C9PKMCYP2C19ALDH1A1
Hydrochloric Acid SCHEMBL27584410 0.99 CYP3A4 (0.52) CYP3A4CYP2C9PKMCYP2C19ALDH1A1
Hydrochloric Acid SCHEMBL7147492 0.99 CYP3A4 (0.52) CYP3A4CYP2C9PKMCYP2C19ALDH1A1
SCHEMBL7102916 0.91 F2 (0.52) CYP3A4CYP2C9PKMCYP2C19ALDH1A1
SCHEMBL21067756 0.89 DPP4 (0.61) CYP3A4CYP2C9PKMCYP2C19ALDH1A1
SCHEMBL21067758 0.89 DPP4 (0.61) CYP3A4CYP2C9PKMCYP2C19ALDH1A1
SCHEMBL27470814 0.87 ALDH1A1 (0.48) CYP3A4CYP2C9PKMCYP2C19ALDH1A1
SCHEMBL7107389 0.87 ALDH1A1 (0.48) CYP3A4CYP2C9PKMCYP2C19ALDH1A1
SCHEMBL7106999 0.86 CYP3A4 (0.58) CYP3A4CYP2C9PKMCYP2C19ALDH1A1
SCHEMBL7102492 0.86 CYP3A4 (0.58) CYP3A4CYP2C9PKMCYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1361212-A1 Peptide derivatives as antithrombotic agents AstraZeneca AB (SE) 2003-11-12 EP claimed
EP-0672658-A1 Antithrombotic agents ELI LILLY AND COMPANY (US) 1995-09-20 EP claimed
WO-1995023609-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 1995-09-08 WO claimed