SCHEMBL7148757

SCHEMBL7148757

C[C@H](N)C(=O)NC(=O)[C@@H]1CC(C2CCCCC2)CN1Cc1ccc(C(N)=NCC(=O)O)nn1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.32
ABCC3 O15438 1/20 0.32
ABCC4 O15439 1/20 0.32
CACNA1F O60840 1/20 0.32
ABCB11 O95342 1/20 0.32
ABCB1 P08183 1/20 0.32
HTR1A P08908 1/20 0.32
DRD2 P14416 1/20 0.32
TACR2 P21452 1/20 0.32
TBXAS1 P24557 1/20 0.32
OPRM1 P35372 1/20 0.32
DRD3 P35462 1/20 0.32
AVPR1A P37288 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
HTR2B P41595 1/20 0.32
CACNA1D Q01668 1/20 0.32
SLC6A3 Q01959 1/20 0.32
KCNH2 Q12809 1/20 0.32
CACNA1S Q13698 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7144856 0.99 CYP3A4 (0.32) CYP3A4ABCC3ABCC4CACNA1FABCB11
SCHEMBL7356317 0.87 F2 (0.37) LMNAUSP2MEN1ACEKMT2A
Hydrochloric Acid SCHEMBL7165069 0.86 F2 (0.37) LMNAUSP2MEN1ACEKMT2A
SCHEMBL7139402 0.84 PTGER4 (0.36) LMNAUSP2MEN1ACEKMT2A
SCHEMBL7143011 0.82 F2 (0.35) CYP3A4LMNAUSP2MEN1ACE
SCHEMBL7148085 0.81 CTSD (0.33) MEN1KMT2A
Hydrochloric Acid SCHEMBL7364149 0.81 F2 (0.34) LMNAUSP2MEN1ACEKMT2A
Hydrochloric Acid SCHEMBL7146333 0.81 CTSD (0.32) MEN1KMT2A
SCHEMBL7249203 0.80 MC3R (0.33) CYP3A4ABCC3ABCC4CACNA1FABCB11
Hydrochloric Acid SCHEMBL7160547 0.80 MC3R (0.33) CYP3A4ABCC3ABCC4CACNA1FABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1361212-A1 Peptide derivatives as antithrombotic agents AstraZeneca AB (SE) 2003-11-12 EP claimed
EP-0672658-A1 Antithrombotic agents ELI LILLY AND COMPANY (US) 1995-09-20 EP claimed
WO-1995023609-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 1995-09-08 WO claimed