SCHEMBL7151125

SCHEMBL7151125

CCc1ccc(-c2nc(N)nc(CCNc3ccc([N+](=O)[O-])c(N)n3)c2-c2cnc[nH]2)cc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.38
MAPT P10636 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
GHSR Q92847 2/20 0.37
NCOA1 Q15788 1/20 0.35
NCOA3 Q9Y6Q9 1/20 0.35
CCNB2 O95067 1/20 0.35
CDK1 P06493 1/20 0.35
CCNB1 P14635 1/20 0.35
GSK3A P49840 1/20 0.35
GSK3B P49841 1/20 0.35
CCNB3 Q8WWL7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7019626 0.81 GSK3B (0.54) CYP2D6MAPTNPSR1NCOA1NCOA3
SCHEMBL4395953 0.80 GSK3B (0.51) MAPTNPSR1CCNB2CDK1CCNB1
SCHEMBL5101039 0.76 GSK3B (0.44) CYP2D6NPSR1GHSRCCNB2CDK1
SCHEMBL7146357 0.71 GSK3B (0.37) CYP2D6NPSR1CCNB2CDK1CCNB1
SCHEMBL2909547 0.69 GSK3B (0.37) CYP2D6CCNB2CDK1CCNB1GSK3A
SCHEMBL4992908 0.69 GSK3B (0.53) MAPTNPSR1CCNB2CDK1CCNB1
Hydrochloric Acid SCHEMBL2911853 0.69 KAT2B (0.37) CYP2D6CCNB2CDK1CCNB1GSK3A
SCHEMBL4395954 0.68 GSK3B (0.69) CYP2D6CCNB2CDK1CCNB1GSK3A
SCHEMBL7025860 0.68 MAPT (0.36) MAPTNPSR1CCNB2CDK1CCNB1
SCHEMBL4393950 0.68 GSK3B (0.50) MAPTNPSR1CCNB2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317433-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2003-06-11 EP disclosed
WO-2002020495-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2002-03-14 WO disclosed
EP-1087963-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 Chiron Corporation (US) 2001-04-04 EP disclosed
WO-1999065897-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 1999-12-23 WO disclosed