SCHEMBL7025860

SCHEMBL7025860

CCc1ccc(C2=C(c3cnc[nH]3)C(Nc3ccc([N+](=O)[O-])c(N)n3)N(CC)C(N)=N2)cc1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CCNB2 O95067 1/20 0.30
CDK1 P06493 1/20 0.30
CCNB1 P14635 1/20 0.30
GSK3A P49840 1/20 0.30
GSK3B P49841 1/20 0.30
CCNB3 Q8WWL7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4395953 0.70 GSK3B (0.51) MAPTNPSR1CCNB2CDK1CCNB1
SCHEMBL7151125 0.68 CYP2D6 (0.38) MAPTNPSR1CCNB2CDK1CCNB1
SCHEMBL5101039 0.63 GSK3B (0.44) NPSR1CCNB2CDK1CCNB1GSK3A
SCHEMBL4393950 0.60 GSK3B (0.50) MAPTNPSR1CCNB2CDK1CCNB1
SCHEMBL4992908 0.60 GSK3B (0.53) MAPTNPSR1CCNB2CDK1CCNB1
SCHEMBL2909547 0.59 GSK3B (0.37) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL27559726 0.59 GSK3B (0.39) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL4395954 0.59 GSK3B (0.69) CCNB2CDK1CCNB1GSK3AGSK3B
Hydrochloric Acid SCHEMBL2911853 0.59 KAT2B (0.37) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL14340675 0.59 ASIC3 (0.68) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317433-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2003-06-11 EP disclosed
WO-2002020495-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2002-03-14 WO disclosed