SCHEMBL715342

SCHEMBL715342

Cc1nc(N)nc(N[C@@H](C)c2cc3cccc(Cl)c3nc2N2CCNC(=O)CC2)n1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 6/20 0.37
PIK3R2 O00459 2/20 0.37
IDH1 O75874 5/20 0.34
PIK3CA P42336 1/20 0.33
MTOR P42345 1/20 0.33
MBOAT4 Q96T53 2/20 0.33
CCNT1 O60563 1/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
CDK9 P50750 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
SOS1 Q07889 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
WEE1 P30291 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL713509 0.92 PIK3CD (0.38) PIK3CDPIK3R2IDH1HRH4SOS1
SCHEMBL713510 0.92 PIK3CD (0.38) PIK3CDPIK3R2IDH1HRH4SOS1
SCHEMBL717467 0.92 PIK3CD (0.41) PIK3CDPIK3CAMTORMBOAT4CCNT1
SCHEMBL714060 0.88 PIK3CD (0.41) PIK3CDIDH1PIK3CAMTOR
SCHEMBL716805 0.84 PIK3CD (0.40) PIK3CDPIK3R2IDH1HRH4SOS1
SCHEMBL15875858 0.84 PIK3CD (0.38) PIK3CDPIK3R2IDH1HRH4SOS1
SCHEMBL716959 0.83 PIK3CB (0.39) PIK3CDPIK3R2PIK3CASOS1
SCHEMBL715439 0.83 CYP1A2 (0.35) PIK3CDPIK3CAMTORMBOAT4CCNT1
SCHEMBL715440 0.83 CYP1A2 (0.35) PIK3CDPIK3CAMTORMBOAT4CCNT1
SCHEMBL17530837 0.83 ADRA2A (0.34) PIK3CDPIK3CAMTORMBOAT4CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2403847-B1 TRIAZINE DERIVATIVES AS KINASE INHIBITORS UCB BIOPHARMA SPRL (BE) 2016-03-02 EP claimed
US-8785628-B2 Triazine derivatives as kinase inhibitors UCB PHARMA, S.A. (BE) 2014-07-22 US claimed
EP-2403847-B1 TRIAZINE DERIVATIVES AS KINASE INHIBITORS UCB BIOPHARMA SPRL (BE) 2016-03-02 EP disclosed
US-8785628-B2 Triazine derivatives as kinase inhibitors UCB PHARMA, S.A. (BE) 2014-07-22 US disclosed
US-20120053167-A1 Triazine Derivatives as Kinase Inhibitors UCB PHARMA, S.A. (BE) 2012-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120053167-A1 Triazine Derivatives as Kinase Inhibitors MAP3K15, PI4KA, MAP3K20 PIK3CD 12/4885PIK3R2 93/4885IDH1 2575/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.