SCHEMBL7157758

SCHEMBL7157758

NC(=O)C1=C/c2ccccc2/N=C/C=C\1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 3/20 0.35
TSHR P16473 2/20 0.32
LMNA P02545 1/20 0.32
MAPK1 P28482 1/20 0.32
SCN4A P35499 1/20 0.32
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32
POLB P06746 1/20 0.31
CYP3A4 P08684 1/20 0.31
PARP1 P09874 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C19 P33261 1/20 0.31
RECQL P46063 1/20 0.31
BLM P54132 1/20 0.31
PMP22 Q01453 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7157768 1.00 TRPA1 (0.35) TRPA1TSHRLMNAMAPK1SCN4A
SCHEMBL19052339 0.70
SCHEMBL17843451 0.66 TRPA1 (0.39) TRPA1TSHRPOLBCYP3A4PARP1
SCHEMBL379612 0.65 TRPA1 (0.33) TRPA1
SCHEMBL379614 0.65 TRPA1 (0.33) TRPA1
SCHEMBL3222323 0.65 TRPA1 (0.41) TRPA1TSHRLMNAMAPK1SCN4A
Fluoride SCHEMBL28557472 0.64 TRPA1 (0.32) TRPA1
SCHEMBL1656527 0.63 TSHR (0.33) TSHRLMNAMAPK1SCN4ASCN5A
SCHEMBL7922049 0.63 TSHR (0.33) TSHRLMNAMAPK1SCN4ASCN5A
SCHEMBL2186647 0.62 KDM4E (0.33) TRPA1LMNAPOLBMAPTRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003014105-A9 BICYCLIC COMPOUND, PRODUCTION AND USE AS HIV INHIBITORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-11-20 WO disclosed