SCHEMBL7159656

SCHEMBL7159656

COc1ccc(-c2cnc3cnccc3c2)cc1OC

nearest known ligand 0.68

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 15/20 0.68
PDGFRA P16234 15/20 0.68
GAK O14976 2/20 0.60
PIK3CD O00329 1/20 0.53
PIK3CA P42336 1/20 0.53
PIK3CB P42338 1/20 0.53
MTOR P42345 1/20 0.53
PIK3CG P48736 1/20 0.53
KDM4E B2RXH2 1/20 0.51
ALDH1A1 P00352 1/20 0.51
HPGD P15428 1/20 0.51
SLC2A1 P11166 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29377512 0.82 PIK3CD (0.73) PDGFRBPDGFRAGAKPIK3CDPIK3CA
SCHEMBL31060782 0.81 PDGFRB (1.00) PDGFRBPDGFRA
SCHEMBL24253008 0.79 MEN1 (0.53) PDGFRBPDGFRAGAKKDM4EALDH1A1
SCHEMBL8500090 0.78 PDGFRB (0.55) PDGFRBPDGFRAPIK3CAKDM4EALDH1A1
Hydrochloric Acid SCHEMBL7162831 0.75 KDM4E (0.65) PDGFRBPDGFRAKDM4EALDH1A1HPGD
SCHEMBL30467740 0.75 PDGFRB (0.44) PDGFRBPDGFRAGAKKDM4EALDH1A1
SCHEMBL24252628 0.75 PDGFRB (0.44) PDGFRBPDGFRAGAKKDM4EALDH1A1
SCHEMBL7153198 0.75 S1PR1 (0.57) PDGFRBPDGFRAGAK
Hydrochloric Acid SCHEMBL7157628 0.74 PDGFRB (0.69) PDGFRBPDGFRAGAKPIK3CDPIK3CA
SCHEMBL26771362 0.74 PDGFRB (0.43) PDGFRBPDGFRAGAKKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030004165-A1 Polyazanaphthalene compounds and pharmaceutical use thereof AJINOMOTO CO. INC (JP) 2003-01-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030004165-A1 Polyazanaphthalene compounds and pharmaceutical use thereof MMP1, TNF, MMP12 PDGFRB 663/4885PDGFRA 1117/4885GAK 1379/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.