Trientine

Trientine

SCHEMBL715994

NCCNCCNCCN.O=S(=O)(O)O

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Trientine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.65
CA6 P23280 5/20 0.65
CA7 P43166 5/20 0.65
CA9 Q16790 5/20 0.65
CA14 Q9ULX7 5/20 0.65
CA5B Q9Y2D0 5/20 0.65
LMNA P02545 4/20 0.65
CA2 P00918 4/20 0.65
CA4 P22748 4/20 0.65
CA5A P35218 4/20 0.65
CA3 P07451 3/20 0.65
ALOX15 P16050 3/20 0.65
TDP1 Q9NUW8 2/20 0.65
CA1 P00915 2/20 0.65
ALDH1A1 P00352 1/20 0.65
TP53 P04637 1/20 0.65
KDM4E B2RXH2 1/20 0.61
MEN1 O00255 2/20 0.59
RECQL P46063 2/20 0.59
KMT2A Q03164 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfuric Acid SCHEMBL8393633 0.97 CA12 (0.62) CA12CA6CA7CA9CA14
Sulfuric Acid SCHEMBL29104260 0.94 CA12 (0.59) CA12CA6CA7CA9CA14
Sulfuric Acid SCHEMBL28250202 0.94 CA12 (0.59) CA12CA6CA7CA9CA14
Sulfuric Acid SCHEMBL11334847 0.94 CA12 (0.59) CA12CA6CA7CA9CA14
Trientine SCHEMBL11114075 0.92 CA6 (0.61) CA12CA6CA7CA9CA14
Sulfamate SCHEMBL18544319 0.92 CA6 (0.61) CA12CA6CA7CA9CA14
Sulfamate SCHEMBL18544358 0.88 CA9 (0.59) CA12CA6CA7CA9CA14
Sulfuric Acid SCHEMBL29044697 0.88 CA12 (0.50) CA12CA6CA7CA9CA14
Sulfuric Acid SCHEMBL17673120 0.87 CA12 (0.50) CA12CA6CA7CA9CA14
Sulfuric Acid SCHEMBL701165 0.87 CA12 (0.50) CA12CA6CA7CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8293673-B2 Process for preparing 4-aminodiphenylamine JIANGSU SINORGCHEM TECHNOLOGY CO., LTD. (CN) 2012-10-23 US claimed
EP-1645555-B1 A METHOD FOR PRODUCING 4-AMINODIPHENYLAMINE JIANGSU SINORGCHEM TECH CO LTD (CN) 2011-09-28 EP claimed
EP-1591438-B1 A PROCESS FOR PREPARING 4-AMINODIPHENYLAMINE SINORGCHEM CO SHANDONG (CN) 2007-11-21 EP claimed
US-20070232832-A1 PROCESS FOR PREPARING 4-AMINODIPHENYLAMINE SINORGCHEM CO. 2007-10-04 US claimed
US-7235694-B2 Reacting nitrobenzene and aniline in presence of a powdery complex base catalyst to perform condensation, hydrogenation, separation and refining; reuse the catalyst; tetraalkyl ammonium hydroxide and a tetraalkyl ammonium salt SINORGCHEM CO., SHANDONG (CN) 2007-06-26 US claimed
US-7176333-B2 Process for preparing 4-aminodiphenylamine SINORGCHEM COMPANY, SHANDONG (CN) 2007-02-13 US claimed
US-7084302-B2 reacting nitrobenzene and aniline in presence of condensation basic catalyst to form mixtures of 4-nitrodiphenylamine and 4-nitrosodiphenylamine, then reacting with hydrogen in the presence of hydrogenation catalysts, separation and refining SINORGCHEM SHANDONG CO., LTD. (CN) 2006-08-01 US claimed
EP-1645555-A1 A METHOD FOR PRODUCING 4-AMINODIPHENYLAMINE Shi, Guangqiang (CN) 2006-04-12 EP claimed
EP-1591438-A1 A PROCESS FOR PREPARING 4-AMINODIPHENYLAMINE Wang, Nongyue (CN) 2005-11-02 EP claimed
US-20050240058-A1 reacting nitrobenzene and aniline in presence of condensation basic catalyst to form mixtures of 4-nitrodiphenylamine and 4-nitrosodiphenylamine, then reacting with hydrogen in the presence of hydrogenation catalysts, separation and refining NONGYUE WANG AND GUANGQIANG SHI (CN) 2005-10-27 US claimed
US-20050065376-A1 Process for preparing 4-aminodiphenylamine GUANGQIANG SHI AND NONGYUE WANG (CN) 2005-03-24 US claimed
CN-116904746-A Recycling treatment method of zinc-containing raw material 北京中金瑞丰环保科技有限公司 2023-10-20 CN disclosed
US-9029603-B2 Process for preparing alkylated p-phenylenediamines JIANGSU SINORGCHEM TECHNOLOGY CO., LTD. (CN) 2015-05-12 US disclosed
US-20130066113-A1 PROCESS FOR PREPARING ALKYLATED P-PHENYLENEDIAMINES JIANGSU SINORGCHEM TECHNOLOGY CO., LTD. (CN) 2013-03-14 US disclosed
US-8293673-B2 Process for preparing 4-aminodiphenylamine JIANGSU SINORGCHEM TECHNOLOGY CO., LTD. (CN) 2012-10-23 US disclosed
US-7084302-B2 reacting nitrobenzene and aniline in presence of condensation basic catalyst to form mixtures of 4-nitrodiphenylamine and 4-nitrosodiphenylamine, then reacting with hydrogen in the presence of hydrogenation catalysts, separation and refining SINORGCHEM SHANDONG CO., LTD. (CN) 2006-08-01 US disclosed
EP-1645555-A1 A METHOD FOR PRODUCING 4-AMINODIPHENYLAMINE Shi, Guangqiang (CN) 2006-04-12 EP disclosed
EP-1591438-A1 A PROCESS FOR PREPARING 4-AMINODIPHENYLAMINE Wang, Nongyue (CN) 2005-11-02 EP disclosed
US-20050240058-A1 reacting nitrobenzene and aniline in presence of condensation basic catalyst to form mixtures of 4-nitrodiphenylamine and 4-nitrosodiphenylamine, then reacting with hydrogen in the presence of hydrogenation catalysts, separation and refining NONGYUE WANG AND GUANGQIANG SHI (CN) 2005-10-27 US disclosed
US-20050065376-A1 Process for preparing 4-aminodiphenylamine GUANGQIANG SHI AND NONGYUE WANG (CN) 2005-03-24 US disclosed