SCHEMBL7160366

SCHEMBL7160366

CCOC(=O)c1onc(OCC)c1CBr

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.45
ALDH1A1 P00352 6/20 0.36
BRD4 O60885 1/20 0.35
BRD2 P25440 1/20 0.35
CREBBP Q92793 1/20 0.35
PKM P14618 2/20 0.35
POLB P06746 2/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
KDM4E B2RXH2 2/20 0.34
CACNA1F O60840 2/20 0.34
CACNA1D Q01668 2/20 0.34
CACNA1S Q13698 2/20 0.34
CACNA1C Q13936 2/20 0.34
TDP2 O95551 2/20 0.34
HTR2C P28335 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7164408 0.88 PLK1 (0.45) PLK1ALDH1A1PKMPOLBLMNA
SCHEMBL7164178 0.81 CYP1A2 (0.40) ALDH1A1BRD4BRD2CREBBPPOLB
SCHEMBL2777897 0.80 PLK1 (0.46) PLK1ALDH1A1PKMPOLBLMNA
SCHEMBL7162885 0.78 GRIA1 (0.56) ALDH1A1MEN1KMT2A
SCHEMBL7162867 0.78 GRIA1 (0.56) ALDH1A1MEN1KMT2A
SCHEMBL7168129 0.73 MAPT (0.43) ALDH1A1HTTNPSR1MEN1KMT2A
SCHEMBL2776180 0.73 GABRA5 (0.54) PLK1ALDH1A1POLBLMNASMN1; SMN2
SCHEMBL2779037 0.72 PLK1 (0.45) PLK1ALDH1A1NPSR1CACNA1FCACNA1D
SCHEMBL2773522 0.72 KDM4E (0.47) PLK1ALDH1A1PKMLMNASMN1; SMN2
SCHEMBL2778352 0.72 PLK1 (0.39) PLK1ALDH1A1PKMPOLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934286-B1 3-ALKOXYISOXAZOL-4-YL-SUBSTITUTED 2-AMINO CARBOXYLIC ACID COMPOUNDS LUNDBECK & CO AS H (DK) 2003-01-08 EP disclosed
US-6200999-B1 ALZHEIMER*S, HUNTINGTON*S, AND PARKINSON*S DISEASE; ANTIEPILEPTIC, ANALGESIC, ANXIOLYTIC, ANTIISCHEMIC AND ANTIDEPRESSANT AGENTS; NMDA AND AMPA RECEPTOR LIGANDS H. LUNDBECK A/S (DK) 2001-03-13 US disclosed
EP-0934286-A1 3-ALKOXYISOXAZOL-4-YL-SUBSTITUTED 2-AMINO CARBOXYLIC ACID COMPOUNDS H. LUNDBECK A/S (DK) 1999-08-11 EP disclosed
WO-1998015542-A1 3-ALKOXYISOXAZOL-4-YL-SUBSTITUTED 2-AMINO CARBOXYLIC ACID COMPOUNDS H. LUNDBECK A/S (DK) 1998-04-16 WO disclosed