SCHEMBL7162249

SCHEMBL7162249

Cc1ccc(Cl)c(Nc2ccccc2)c1Cl

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.58
MEN1 O00255 2/20 0.58
MAPK1 P28482 2/20 0.58
KMT2A Q03164 2/20 0.58
METTL3 Q86U44 2/20 0.58
AKR1B10 O60218 1/20 0.58
ABCB11 O95342 1/20 0.58
TTR P02766 1/20 0.58
ADORA3 P0DMS8 1/20 0.58
CHRM1 P11229 1/20 0.58
FABP2 P12104 1/20 0.58
RXRA P19793 1/20 0.58
TBXA2R P21731 1/20 0.58
NR4A1 P22736 1/20 0.58
PTGS1 P23219 1/20 0.58
PDE4A P27815 1/20 0.58
AKR1C3 P42330 1/20 0.58
NR4A2 P43354 1/20 0.58
AKR1C2 P52895 1/20 0.58
AKR1C1 Q04828 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9735867 0.83 PTGS2 (0.53) PTGS2MEN1MAPK1KMT2AMETTL3
SCHEMBL24021583 0.80 PTGS2 (0.57) PTGS2MEN1MAPK1KMT2AMETTL3
SCHEMBL8611927 0.80 PTGS2 (0.44) PTGS2MEN1MAPK1KMT2AMETTL3
SCHEMBL2760397 0.79 PTGS2 (0.65) PTGS2MEN1MAPK1KMT2AMETTL3
SCHEMBL24021602 0.78 MEN1 (0.56) PTGS2MEN1MAPK1KMT2AMETTL3
SCHEMBL14618510 0.78 PTGS2 (0.53) PTGS2MEN1MAPK1KMT2APTGS1
SCHEMBL8611985 0.77 PTGS2 (0.42) PTGS2MEN1MAPK1KMT2AMETTL3
SCHEMBL22140749 0.77 CLCN2 (0.62) PTGS2MEN1MAPK1KMT2AMETTL3
SCHEMBL20694079 0.75 PTGS2 (0.60) PTGS2MEN1MAPK1KMT2AMETTL3
SCHEMBL2419050 0.74 HSD17B10 (0.52) PTGS2MEN1MAPK1KMT2AAKR1B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2409149-B1 METHODS OF SCREENING USING AMPHIBIANS BRÄNDLI ANDRÉ W (CH) 2015-11-11 EP disclosed
US-6552077-B2 Kidney disorders EXOCELL, INC. 2003-04-22 US disclosed
EP-1242069-A2 ALBUMIN-BINDING COMPOUNDS THAT PREVENT NONENZYMATIC GLYCATION AND THAT MAY BE USED FOR TREATMENT OF GLYCATION-RELATED PATHOLOGIES EXOCELL, INC. (US) 2002-09-25 EP disclosed
US-6355680-B1 BLOCKING REACTION OF GLUCOSE AND ALBUMIN EXOCELL, INC. 2002-03-12 US disclosed
US-20010034359-A1 Albumin-binding compounds that prevent nonenzymatic glycation and that may be used for treatment of glycation-related pathologies EXOCELL, INC. 2001-10-25 US disclosed
WO-2001003684-A2 ALBUMIN-BINDING COMPOUNDS THAT PREVENT NONENZYMATIC GLYCATION AND THAT MAY BE USED FOR TREATMENT OF GLYCATION-RELATED PATHOLOGIES EXOCELL, INC. (US) 2001-01-18 WO disclosed
US-5462952-A Have activity as inhibitors of 5-lipoxygenase and/or cyclooxygenase WARNER-LAMBERT COMPANY (US) 1995-10-31 US disclosed
US-5155110-A Antiinflammatory agents, analgesics, antipyretics WARNER-LAMBERT COMPANY (US) 1992-10-13 US disclosed
EP-0316630-A1 Novel fenamic acid hydroxamate derivatives having cyclooxygenase and 5-lipoxygenase inhibition WARNER-LAMBERT COMPANY (US) 1989-05-24 EP disclosed
WO-1989003818-A1 NOVEL FENAMIC ACID HYDROXAMATE DERIVATIVES HAVING CYCLOOXYGENASE AND 5-LIPOXYGENASE INHIBITION WARNER-LAMBERT COMPANY (US) 1989-05-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010034359-A1 Albumin-binding compounds that prevent nonenzymatic glycation and that may be used for treatment of glycation-related pathologies ALB, AGER, TTR PTGS2 2067/4885MEN1 3564/4885MAPK1 2536/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.