SCHEMBL7162502

SCHEMBL7162502

C=CCc1nc2c(c(=O)[nH]1)CNCC2

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.46
TNKS O95271 1/20 0.37
TNKS2 Q9H2K2 1/20 0.37
CHRM3 P20309 1/20 0.33
NPSR1 Q6W5P4 1/20 0.31
PARP1 P09874 1/20 0.31
HTR2A P28223 1/20 0.30
HTR2B P41595 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227586 0.80 HTR2C (0.49) HTR2CTNKSTNKS2PARP1HTR2A
SCHEMBL7162498 0.77 PARP1 (0.37) CHRM3PARP1
SCHEMBL31351621 0.71 HTR2C (0.63) HTR2CTNKSTNKS2HTR2AHTR2B
SCHEMBL25431342 0.71 HPGD (0.41) HTR2CTNKSTNKS2CHRM3PARP1
SCHEMBL23972783 0.69 HTR2C (0.56) HTR2CTNKSTNKS2PARP1
SCHEMBL5228377 0.68 HTR2C (0.49) HTR2CTNKSTNKS2PARP1HTR2B
SCHEMBL14344503 0.65 MTHFD2 (0.49) HTR2CTNKSTNKS2PARP1HTR2A
SCHEMBL9232984 0.65 ALDH1A1 (0.32) NPSR1
SCHEMBL23973135 0.62 HTR2C (0.51) HTR2CTNKSTNKS2PARP1HTR2A
SCHEMBL23972240 0.61 TNKS (0.47) HTR2CTNKSTNKS2PARP1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6638937-B2 As antihypertensive agents; for therapy of disorders related to renal, glomerular and mesangial cell function; therapy of endotoxemia or endotoxin shock as well as hemorrhagic shock; useful in alleviation of pain associated cancer BRISTOL-MYERS SQUIBB CO. 2003-10-28 US disclosed