SCHEMBL7166205

SCHEMBL7166205

[AsH2][C@@H]1COc2ccccc2SC1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.38
DAO P14920 1/20 0.37
SCN5A Q14524 1/20 0.37
LMNA P02545 2/20 0.33
CRHBP P24387 2/20 0.33
CRHR2 Q13324 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
HTT P42858 1/20 0.33
OXTR P30559 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
ITGB2 P05107 1/20 0.32
ICAM1 P05362 1/20 0.32
ITGAL P20701 1/20 0.32
CYP19A1 P11511 1/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7166201 1.00 NISCH (0.38) NISCHDAOSCN5ALMNACRHBP
SCHEMBL2069021 0.78 NISCH (0.39) NISCHDAOSCN5AALDH1A1HPGD
SCHEMBL6069296 0.78 NISCH (0.39) NISCHDAOSCN5AALDH1A1HPGD
SCHEMBL2071541 0.78 NISCH (0.39) NISCHDAOSCN5AALDH1A1HPGD
SCHEMBL57996 0.69
SCHEMBL29395105 0.69
SCHEMBL255962 0.67 ITGB2 (0.52) LMNACRHBPCRHR2SMN1; SMN2ALDH1A1
SCHEMBL29395580 0.67 ITGB2 (0.52) LMNACRHBPCRHR2SMN1; SMN2ALDH1A1
SCHEMBL6097642 0.66 ADRA1A (0.45) NISCHHTTMEN1KMT2A
SCHEMBL24214454 0.65 NISCH (0.46) NISCHSCN5ALMNASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1370547-A1 BENZOAXATHIEPIN DERIVATIVES AND THEIR USE AS MEDICINES PIERRE FABRE MEDICAMENT (FR) 2003-12-17 EP disclosed
WO-2002081464-A1 BENZOAXATHIEPIN DERIVATIVES AND THEIR USE AS MEDICINES PIERRE FABRE MEDICAMENT (FR) 2002-10-17 WO disclosed