SCHEMBL7167161

SCHEMBL7167161

CCOC(=O)CC[C@@H](NC(=O)c1ccc([N+](=O)[O-])c(C)c1)C(=O)OCC

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.53
ALDH1A1 P00352 2/20 0.53
HPGD P15428 2/20 0.53
KDM4E B2RXH2 1/20 0.53
HSD17B10 Q99714 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
MAPT P10636 1/20 0.53
KMT2A Q03164 5/20 0.49
POLB P06746 3/20 0.49
LMNA P02545 1/20 0.48
TSHR P16473 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
GAA P10253 3/20 0.46
MEN1 O00255 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7167160 1.00 L3MBTL1 (0.53) L3MBTL1ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL27286692 1.00 L3MBTL1 (0.53) L3MBTL1ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL9782310 0.89 ALDH1A1 (0.52) L3MBTL1ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL9782307 0.89 ALDH1A1 (0.52) L3MBTL1ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL9782445 0.89 ALDH1A1 (0.51) L3MBTL1ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL9782435 0.89 ALDH1A1 (0.51) L3MBTL1ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL31389132 0.85 L3MBTL1 (0.61) L3MBTL1ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL7954572 0.84 ALDH1A1 (0.55) L3MBTL1ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL7775216 0.84 ALDH1A1 (0.55) L3MBTL1ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL7954574 0.84 ALDH1A1 (0.55) L3MBTL1ALDH1A1HPGDKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6559149-B1 Lesser side effects without compromise in their efficacy CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-05-06 US disclosed
EP-0632038-B1 METHOTREXATE DERIVATIVE CHUGAI PHARMACEUTICAL CO LTD (JP) 2001-08-22 EP disclosed
CN-1039907-C Methotrexate derivative CHUGAI PHARMACEUTICAL CO LTD (JP) 1998-09-23 CN disclosed
EP-0632038-A1 METHOTREXATE DERIVATIVE Chugai Seiyaku Kabushiki Kaisha (JP) 1995-01-04 EP disclosed
CN-1077956-A METHOTREXATE DERIVATIVE CHUGAI PHARMACEUTICAL CO LTD (JP) 1993-11-03 CN disclosed
US-5019577-A Novel compounds and use BURROUGHS WELCOME CO. (US) 1991-05-28 US disclosed