SCHEMBL7170258

SCHEMBL7170258

COc1ccc(C2(C)CCC(=O)O2)cc1OC1CCCC1

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 19/20 0.60
PDE4A P27815 19/20 0.60
PDE4C Q08493 18/20 0.60
PDE4D Q08499 18/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7178980 1.00 PDE4B (0.60) PDE4BPDE4APDE4CPDE4D
SCHEMBL7170256 1.00 PDE4B (0.60) PDE4BPDE4APDE4CPDE4D
SCHEMBL7174439 0.98 PDE4B (0.57) PDE4BPDE4APDE4CPDE4D
SCHEMBL7175034 0.98 PDE4B (0.57) PDE4BPDE4APDE4CPDE4D
SCHEMBL7171569 0.98 PDE4B (0.57) PDE4BPDE4APDE4CPDE4D
SCHEMBL7172425 0.86 LMNA (0.48) PDE4BPDE4APDE4CPDE4D
SCHEMBL7172429 0.86 LMNA (0.48) PDE4BPDE4APDE4CPDE4D
SCHEMBL6585386 0.84 PDE4A (0.56) PDE4BPDE4APDE4CPDE4D
SCHEMBL6585249 0.83 PDE4B (0.56) PDE4BPDE4APDE4CPDE4D
SCHEMBL7176094 0.83 PDE4B (0.57) PDE4BPDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900212-B1 CHIRAL PHENYLDIHYDROFURANONES AS PDE-IV INHIBITORS SCHERING AG (DE) 2003-12-17 EP claimed
US-6011060-A TREATING A DISEASE MEDIATED BY ACTIVATION OF THE TUMOR NECROSIS FACTOR SCHERING AKTIENGESELLSCHAFT (DE) 2000-01-04 US claimed
EP-0900212-B1 CHIRAL PHENYLDIHYDROFURANONES AS PDE-IV INHIBITORS SCHERING AG (DE) 2003-12-17 EP disclosed
US-6011060-A TREATING A DISEASE MEDIATED BY ACTIVATION OF THE TUMOR NECROSIS FACTOR SCHERING AKTIENGESELLSCHAFT (DE) 2000-01-04 US disclosed
EP-0900212-A1 CHIRAL PHENYLDIHYDROFURANONES AS PDE-IV INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1999-03-10 EP disclosed
WO-1997040032-A1 CHIRAL PHENYLDIHYDROFURANONES AS PDE-IV INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-10-30 WO disclosed