SCHEMBL7175691

SCHEMBL7175691

Nc1c(Cl)cc(C(F)(F)F)cc1NC(=S)Nc1ccc(NC(=O)c2ccco2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.54
NPSR1 Q6W5P4 4/20 0.54
MEN1 O00255 4/20 0.54
HTT P42858 1/20 0.54
USP2 O75604 1/20 0.52
TSHR P16473 1/20 0.52
RAB9A P51151 5/20 0.49
NPC1 O15118 4/20 0.49
CASP3 P42574 1/20 0.49
SENP8 Q96LD8 1/20 0.49
SENP7 Q9BQF6 1/20 0.49
SENP6 Q9GZR1 1/20 0.49
ALDH1A1 P00352 6/20 0.47
KDM4E B2RXH2 2/20 0.47
GFER P55789 1/20 0.47
AHR P35869 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
MAPT P10636 6/20 0.47
POLB P06746 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6816683 0.80 ALDH1A1 (0.52) KMT2ANPSR1MEN1HTTRAB9A
SCHEMBL6816676 0.80 ALDH1A1 (0.46) KMT2ANPSR1MEN1ALDH1A1KDM4E
SCHEMBL6815053 0.79 MAPT (0.60) KMT2ANPSR1MEN1RAB9ANPC1
SCHEMBL7162313 0.79 MEN1 (0.86) KMT2ANPSR1MEN1HTTUSP2
SCHEMBL7778713 0.76 RAB9A (0.67) KMT2ANPSR1MEN1HTTRAB9A
SCHEMBL7848327 0.74 RAB9A (0.69) KMT2AMEN1RAB9ANPC1CASP3
SCHEMBL7157873 0.74 NPSR1 (0.55) KMT2ANPSR1MEN1HTTUSP2
SCHEMBL7163720 0.74 MEN1 (0.60) KMT2ANPSR1MEN1HTTUSP2
SCHEMBL7162970 0.74 MYC (0.65) KMT2ANPSR1MEN1HTTUSP2
SCHEMBL7848400 0.73 RAB9A (0.66) KMT2ANPSR1MEN1HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6555561-B2 N-(5-((((5-Chloro-2,4-dimethoxyphenyl)amino)thioxomethyl)-amino)-2 -pyridinyl)-2-methylbenzamide, for example; inhibiting replication of a herpes virus WYETH 2003-04-29 US disclosed