SCHEMBL7180856

SCHEMBL7180856

CCOC(=O)C(C)CCC1CCN(CC(=O)c2ccc3c(c2)N(COC)c2nccnc2S3)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ICAM1 P05362 6/20 0.42
HDAC6 Q9UBN7 2/20 0.35
CHRM2 P08172 2/20 0.35
HTR1A P08908 2/20 0.35
CHRM1 P11229 2/20 0.35
DRD2 P14416 2/20 0.35
ADRA2B P18089 2/20 0.35
ADRA2C P18825 2/20 0.35
CHRM3 P20309 2/20 0.35
HTR2A P28223 2/20 0.35
HTR2C P28335 2/20 0.35
ADRA1A P35348 2/20 0.35
HRH1 P35367 2/20 0.35
DRD3 P35462 2/20 0.35
OPRK1 P41145 2/20 0.35
HTR2B P41595 2/20 0.35
KCNH2 Q12809 2/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7173360 0.87 ICAM1 (0.45) ICAM1HDAC6CHRM2HTR1ACHRM1
SCHEMBL8522771 0.83 ICAM1 (0.43) ICAM1HDAC6CHRM2HTR1ACHRM1
SCHEMBL6746537 0.82 ICAM1 (0.41) ICAM1HDAC6MEN1KMT2AALDH1A1
SCHEMBL8522768 0.81 ICAM1 (0.36) ICAM1HDAC6CHRM2HTR1ACHRM1
SCHEMBL6745590 0.80 ICAM1 (0.64) ICAM1
SCHEMBL7149885 0.76 ICAM1 (0.53) ICAM1MEN1KMT2AALDH1A1FAAH
SCHEMBL7144340 0.73 HDAC6 (0.42) HDAC6CHRM2HTR1ACHRM1DRD2
SCHEMBL8315505 0.73 HDAC6 (0.45) HDAC6CHRM2HTR1ACHRM1DRD2
SCHEMBL6745150 0.72 HDAC6 (0.44) HDAC6CHRM2HTR1ACHRM1DRD2
SCHEMBL6751888 0.72 ICAM1 (0.43) ICAM1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6518423-B1 These compounds are useful as drugs efficacious in the prevention and treatment of these various inflammatory diseases and immunologic diseases, such as rheumatoid arthritis, atopic dermatitis, psoriasis, asthma, and EISAI CO., LTD. (JP) 2003-02-11 US disclosed
EP-0934941-A1 BENZOPIPERIDINE DERIVATIVES Eisai Co., Ltd. (JP) 1999-08-11 EP disclosed