SCHEMBL7181745

SCHEMBL7181745

C=CC(=O)/C=C/c1ccncc1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JUN P05412 2/20 0.77
NFKB1 P19838 2/20 0.77
MAPT P10636 4/20 0.47
KDM4E B2RXH2 2/20 0.47
NPC1 O15118 1/20 0.47
MAPK1 P28482 1/20 0.47
RAB9A P51151 1/20 0.47
GPR55 Q9Y2T6 1/20 0.47
CYP1A2 P05177 6/20 0.47
CYP2D6 P10635 3/20 0.47
ALDH1A1 P00352 3/20 0.47
F3 P13726 3/20 0.47
CYP2C9 P11712 2/20 0.47
PLIN1 O60240 1/20 0.47
LMNA P02545 1/20 0.47
RECQL P46063 1/20 0.47
PLIN5 Q00G26 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
ABHD5 Q8WTS1 1/20 0.47
KDM1A O60341 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7181746 1.00 JUN (0.77) JUNNFKB1MAPTKDM4ENPC1
SCHEMBL5598760 0.87 JUN (1.00) JUNNFKB1MAPTKDM4ENPC1
SCHEMBL5598762 0.87 JUN (1.00) JUNNFKB1MAPTKDM4ENPC1
Hydrochloric Acid SCHEMBL11970821 0.85 JUN (0.95) JUNNFKB1MAPTKDM4ENPC1
Hydrochloric Acid SCHEMBL11970816 0.85 JUN (0.95) JUNNFKB1MAPTKDM4ENPC1
SCHEMBL11999793 0.80 JUN (0.84) JUNNFKB1MAPTKDM4ENPC1
SCHEMBL4421926 0.79 MAPT (0.75) MAPTNPC1CYP1A2CYP2D6ALDH1A1
SCHEMBL184544 0.79 MAPT (0.75) MAPTNPC1CYP1A2CYP2D6ALDH1A1
Hydrochloric Acid SCHEMBL1490918 0.78 JUN (0.81) JUNNFKB1MAPTKDM4ENPC1
Hydrochloric Acid SCHEMBL1490919 0.78 JUN (0.81) JUNNFKB1MAPTKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946190-B1 METHODS AND COMPOSITIONS FOR STIMULATING NEURITE OUTGROWTH VERTEX PHARMA (US) 2003-09-24 EP disclosed
EP-0946190-A1 METHODS AND COMPOSITIONS FOR STIMULATING NEURITE GROWTH USING COMPOUNDS WITH AFFINITY FOR FKBP12 IN COMBINATION WITH NEUROTROPHIC FACTORS Vertex Pharmaceuticals Incorporated (US) 1999-10-06 EP disclosed
WO-1998020891-A1 METHODS AND COMPOSITIONS FOR STIMULATING NEURITE GROWTH USING COMPOUNDS WITH AFFINITY FOR FKBP12 IN COMBINATION WITH NEUROTROPHIC FACTORS VERTEX PHARMACEUTICALS INCORPORATED (US) 1998-05-22 WO disclosed