SCHEMBL7182817

SCHEMBL7182817

CCN(CC)C(=O)C=Cc1ccc(Oc2c(-c3ccc(O)cc3)ccc3ccccc23)cc1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 13/20 0.51
ESR2 Q92731 13/20 0.51
NPC1 O15118 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
LTB4R Q15722 1/20 0.47
LTB4R2 Q9NPC1 1/20 0.47
BACE1 P56817 3/20 0.43
ABCG2 Q9UNQ0 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7195408 0.92 ESR1 (0.51) ESR1ESR2NPC1L3MBTL1LTB4R
SCHEMBL7187504 0.85 CA12 (0.56) ESR1ESR2BACE1
SCHEMBL7182549 0.84 ESR1 (0.60) ESR1ESR2
SCHEMBL7182543 0.84 ESR1 (0.60) ESR1ESR2
SCHEMBL7189415 0.81 ESR1 (0.48) ESR1ESR2BACE1
SCHEMBL7189412 0.81 ESR1 (0.48) ESR1ESR2BACE1
SCHEMBL7190060 0.79 ESR1 (0.40) ESR1ESR2NPC1LTB4R2
SCHEMBL7189519 0.79 ESR1 (0.54) ESR1ESR2
SCHEMBL7189979 0.78 ESR1 (0.51) ESR1ESR2NPC1
SCHEMBL7183993 0.78 ESR1 (0.59) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0835867-B1 1-Aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods LILLY CO ELI (US) 2003-12-03 EP claimed