SCHEMBL7183175

SCHEMBL7183175

N#Cc1ccccc1CS(=O)(=O)[C@H](CNC(=O)C1CCNCC1)C(=O)NCCC(C(=O)c1nc2ccccc2o1)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSS P25774 18/20 0.39
CTSL P07711 2/20 0.39
CTSB P07858 2/20 0.39
CTSK P43235 2/20 0.39
LMNA P02545 2/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6463875 1.00 CTSS (0.39) CTSSCTSLCTSBCTSKLMNA
SCHEMBL6062088 0.94 CTSS (0.36) CTSSCTSLCTSBCTSKLMNA
SCHEMBL7048383 0.91 LMNA (0.40) CTSSLMNAHTTSMN1; SMN2CYP3A4
SCHEMBL6467213 0.87 LMNA (0.38) CTSSLMNAHTTSMN1; SMN2CYP3A4
SCHEMBL7044345 0.85 CTSS (0.39) CTSSCTSLCTSBCTSKLMNA
SCHEMBL7042145 0.84 CTSS (0.40) CTSSCTSLCTSBCTSKLMNA
SCHEMBL6062750 0.83 EPHX2 (0.38) CTSSLMNAHTTCYP3A4CYP2C9
SCHEMBL6464521 0.80 CTSS (0.38) CTSSCTSLCTSKLMNAHTT
SCHEMBL7183010 0.79 CTSS (0.37) CTSSLMNAHTTSMN1; SMN2CYP3A4
SCHEMBL7042876 0.79 CTSS (0.43) CTSSCTSLCTSBCTSKLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6576630-B1 Alkanoyl substituted benzooxazoles or naphthooxazoles AXYS PHARMACEUTICALS, INC. 2003-06-10 US disclosed