SCHEMBL7183324

SCHEMBL7183324

CC(C)(C)OC(=O)N1C=CC=Nc2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.43
KDM1A O60341 1/20 0.38
GRM5 P41594 2/20 0.34
GRM1 Q13255 2/20 0.34
GPR119 Q8TDV5 2/20 0.33
SCN9A Q15858 2/20 0.33
SCN5A Q14524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
MAPK1 P28482 1/20 0.33
SMARCA2 P51531 1/20 0.32
SMARCA4 P51532 1/20 0.32
PBRM1 Q86U86 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CYP11B2 P19099 1/20 0.32
CKS1B P61024 1/20 0.32
SKP1 P63208 1/20 0.32
SKP2 Q13309 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5172363 0.74 BCHE (0.46) BCHEKDM1AGRM5GRM1GPR119
SCHEMBL27928991 0.70 BCHE (0.44) BCHEKDM1AGRM5GRM1GPR119
SCHEMBL4253863 0.70 BCHE (0.57) BCHEKDM1AGPR119MAPK1
SCHEMBL6255939 0.69 BCHE (0.46) BCHEKDM1AGPR119HDAC1HDAC6
SCHEMBL5670700 0.69 BCHE (0.46) BCHEKDM1AGRM5GRM1GPR119
SCHEMBL38658293 0.69 BCHE (0.46) BCHEKDM1AGRM5GRM1GPR119
SCHEMBL3459528 0.65 BCHE (0.48) BCHEKDM1AGPR119HDAC1HDAC6
SCHEMBL7020597 0.65 BCHE (0.44) BCHEKDM1AGRM5GRM1GPR119
SCHEMBL9655258 0.64 KDM4E (0.46) MEN1KMT2A
SCHEMBL6994927 0.64 BCHE (0.43) BCHEKDM1AGRM5GRM1GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003031376-A1 SOLID PHASE SYNTHESIS OF SUBSTITUTED 1,5-BENZODIAZEPINE-2-ONE AND 1,5-BENZOTHIAZEPINE-2-ONE AVENTIS PHARMACEUTICALS INC. (US) 2003-04-17 WO disclosed