SCHEMBL7183476

SCHEMBL7183476

CC(C)(C)OC(=O)N[C@H]1CC[C@H](Nc2ccc(C(F)(F)F)cc2[N+](=O)[O-])CC1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.55
MAPK1 P28482 6/20 0.53
NPSR1 Q6W5P4 1/20 0.52
HCAR3 P49019 3/20 0.50
STAT3 P40763 1/20 0.47
MAPT P10636 4/20 0.47
ALDH1A1 P00352 2/20 0.47
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
AKR1B1 P15121 1/20 0.45
AKR1C4 P17516 1/20 0.45
AKR1C3 P42330 1/20 0.45
AKR1C2 P52895 1/20 0.45
AKR1C1 Q04828 1/20 0.45
KCNMA1 Q12791 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7183491 1.00 PKM (0.55) PKMMAPK1NPSR1HCAR3STAT3
SCHEMBL1015485 0.86 HCAR3 (0.53) HCAR3MAPTALDH1A1MEN1KMT2A
SCHEMBL1015486 0.86 HCAR3 (0.53) HCAR3MAPTALDH1A1MEN1KMT2A
SCHEMBL16989691 0.85 HCAR3 (0.52) PKMMAPK1HCAR3MAPTALDH1A1
SCHEMBL15599592 0.85 HCAR3 (0.52) PKMMAPK1HCAR3MAPTALDH1A1
SCHEMBL2860350 0.84 MAPK1 (0.58) PKMMAPK1NPSR1HCAR3STAT3
SCHEMBL18687361 0.83 HCAR3 (0.50) MAPK1NPSR1HCAR3MAPTALDH1A1
SCHEMBL4437146 0.82 MAPT (0.64) MAPK1NPSR1MAPTALDH1A1MEN1
SCHEMBL7177008 0.82 HCAR3 (0.49) HCAR3MAPTMEN1KMT2A
SCHEMBL7176994 0.82 HCAR3 (0.49) HCAR3MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6582351-B1 Benzimidazole heterocyclic compounds having pharmacological activities, and their use as a medicament for treatment or prevention of diseases mediated by cGMP-PDE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-06-24 US disclosed