SCHEMBL7183957

SCHEMBL7183957

O=CNC1CCC(n2c(=O)[nH]c3cc(C(F)(F)F)ccc32)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
OPRM1 P35372 2/20 0.48
HSD11B1 P28845 2/20 0.45
SIRT2 Q8IXJ6 1/20 0.44
TNKS O95271 1/20 0.43
PARP1 P09874 1/20 0.43
PARP2 Q9UGN5 1/20 0.43
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
HSP90AA1 P07900 1/20 0.43
CYP3A4 P08684 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43
CYP2C19 P33261 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7183953 1.00 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2OPRM1HSD11B1SIRT2
SCHEMBL7179611 0.82 ALDH1A1 (0.62) ALDH1A1SMN1; SMN2OPRM1HSD11B1SIRT2
SCHEMBL7179604 0.82 ALDH1A1 (0.62) ALDH1A1SMN1; SMN2OPRM1HSD11B1SIRT2
SCHEMBL7191677 0.82 ALDH1A1 (0.61) ALDH1A1SMN1; SMN2OPRM1HSD11B1SIRT2
SCHEMBL4750867 0.81 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2OPRM1HSD11B1SIRT2
SCHEMBL31285855 0.81 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2OPRM1HSD11B1SIRT2
SCHEMBL7178523 0.80 JAK2 (0.39) ALDH1A1SMN1; SMN2OPRM1HSD11B1TNKS
SCHEMBL7178530 0.80 JAK2 (0.39) ALDH1A1SMN1; SMN2OPRM1HSD11B1TNKS
SCHEMBL7185917 0.80 ALDH1A1 (0.59) ALDH1A1SMN1; SMN2OPRM1HSD11B1SIRT2
SCHEMBL7184352 0.80 TNKS (0.54) OPRM1HSD11B1SIRT2TNKSPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6582351-B1 Benzimidazole heterocyclic compounds having pharmacological activities, and their use as a medicament for treatment or prevention of diseases mediated by cGMP-PDE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-06-24 US disclosed