SCHEMBL7185041

SCHEMBL7185041

CC=CCc1cc(C=CC(=O)c2ccc(NC)cc2)c(OC(C)C)c(CC=CC)c1O

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 12/20 0.36
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CYP3A4 P08684 1/20 0.35
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7185037 1.00 PTPN1 (0.36) PTPN1CTSLCTSBCYP3A4ALDH1A1
SCHEMBL7190654 0.90 PTPN1 (0.44) PTPN1CTSLCTSB
SCHEMBL7190659 0.90 PTPN1 (0.44) PTPN1CTSLCTSB
SCHEMBL7190370 0.89 CTSL (0.43) PTPN1CTSLCTSBCYP3A4ALDH1A1
SCHEMBL7190096 0.89 PTPN1 (0.44) PTPN1CTSLCTSBALDH1A1LMNA
SCHEMBL7190102 0.89 PTPN1 (0.44) PTPN1CTSLCTSBALDH1A1LMNA
SCHEMBL7190368 0.89 CTSL (0.43) PTPN1CTSLCTSBCYP3A4ALDH1A1
SCHEMBL7186294 0.87 PTPN1 (0.47) PTPN1
SCHEMBL7186296 0.87 PTPN1 (0.47) PTPN1
SCHEMBL7190903 0.87 PTPN1 (0.41) PTPN1ALDH1A1LMNAMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP disclosed
US-5985935-A PARASITICIDES OR BACTERICIDES STATENS SERUMINSTITUT (DK) 1999-11-16 US disclosed