SCHEMBL7190096

SCHEMBL7190096

C/C=C/Cc1cc(/C=C/C(=O)c2ccc(NC)cc2)c(OC)c(C/C=C/C)c1O

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 9/20 0.44
CTSL P07711 3/20 0.41
CTSB P07858 3/20 0.41
ABCG2 Q9UNQ0 2/20 0.40
CAPN1 P07384 1/20 0.39
GABRA3 P34903 1/20 0.39
GABRA2 P47869 1/20 0.39
GABRB2 P47870 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MAPT P10636 2/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7190102 1.00 PTPN1 (0.44) PTPN1CTSLCTSBABCG2CAPN1
SCHEMBL7190901 0.90 PTPN1 (0.41) PTPN1ABCG2MAPTALDH1A1LMNA
SCHEMBL7190903 0.90 PTPN1 (0.41) PTPN1ABCG2MAPTALDH1A1LMNA
SCHEMBL7180300 0.89 PTPN1 (0.54) PTPN1CTSLCTSBABCG2CAPN1
SCHEMBL7180303 0.89 PTPN1 (0.54) PTPN1CTSLCTSBABCG2CAPN1
SCHEMBL7185037 0.89 PTPN1 (0.36) PTPN1CTSLCTSBMAPTALDH1A1
SCHEMBL7185041 0.89 PTPN1 (0.36) PTPN1CTSLCTSBMAPTALDH1A1
SCHEMBL7178908 0.89 CTSL (0.51) PTPN1CTSLCTSBABCG2CAPN1
SCHEMBL7178910 0.89 CTSL (0.51) PTPN1CTSLCTSBABCG2CAPN1
SCHEMBL7184617 0.88 DPP4 (0.39) PTPN1CTSLCTSBABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP disclosed
US-5985935-A PARASITICIDES OR BACTERICIDES STATENS SERUMINSTITUT (DK) 1999-11-16 US disclosed