SCHEMBL7185408

SCHEMBL7185408

Cc1ccc(-n2c[c]nc2C)cc1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALKBH5 Q6P6C2 1/20 0.39
NOTUM Q6P988 4/20 0.37
FLT1 P17948 1/20 0.34
KDR P35968 1/20 0.34
S1PR1 P21453 3/20 0.33
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
HSD11B1 P28845 2/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31
AR P10275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7160454 0.73 ALKBH5 (0.39) ALKBH5NOTUMFLT1KDRS1PR1
SCHEMBL7155610 0.71 POLB (0.48)
SCHEMBL7254837 0.70 AR (0.41) AR
SCHEMBL16181625 0.67 AR (0.53) ALKBH5NOTUMPDE3BPDE3AHTR2A
SCHEMBL16181629 0.67 AR (0.53) ALKBH5NOTUMPDE3BPDE3AHTR2A
SCHEMBL13122994 0.66 AR (0.49) ALKBH5NOTUMHTR2AHTR2CHTR2B
SCHEMBL28166708 0.65 AR (0.48) ALKBH5NOTUMHTR2AHTR2CHTR2B
SCHEMBL13122748 0.65 CYP3A4 (0.50) NOTUMPDE3BPDE3A
SCHEMBL13122732 0.65 PDK2 (0.46) ALKBH5NOTUMFLT1KDRHSD11B1
SCHEMBL13485858 0.64 COMT (0.56) ALKBH5NOTUMFLT1KDRPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358165-A1 IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-11-05 EP disclosed
WO-2002060877-A1 IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-08-08 WO disclosed