SCHEMBL7186268

SCHEMBL7186268

O=C(O)c1nccn1Cc1ccc(F)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.67
NPC1 O15118 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
LMNA P02545 1/20 0.50
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
TP53 P04637 2/20 0.45
OPRD1 P41143 2/20 0.44
OPRK1 P41145 1/20 0.44
KDM4A O75164 1/20 0.44
KDM5A P29375 1/20 0.44
KDM4C Q9H3R0 1/20 0.44
KDM5B Q9UGL1 1/20 0.44
MAPT P10636 1/20 0.44
THRB P10828 1/20 0.44
HSP90AA1 P07900 1/20 0.44
HSP90B1 P14625 1/20 0.44
CNR2 P34972 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lithium SCHEMBL7185471 0.98 RAB9A (0.66) RAB9ANPC1SMN1; SMN2LMNACA12
SCHEMBL28413277 0.86 RAB9A (0.51) RAB9ANPC1SMN1; SMN2OPRD1OPRK1
SCHEMBL12803743 0.86 SMN1; SMN2 (0.51) RAB9ANPC1SMN1; SMN2LMNAHSP90AA1
SCHEMBL418384 0.85 RAB9A (0.57) RAB9ANPC1SMN1; SMN2OPRD1OPRK1
SCHEMBL28418521 0.84 RAB9A (0.50) RAB9ANPC1SMN1; SMN2
SCHEMBL28419096 0.84 RAB9A (0.50) RAB9ANPC1SMN1; SMN2
SCHEMBL28413304 0.84 RAB9A (0.67) RAB9ANPC1SMN1; SMN2LMNATP53
Hydrochloric Acid SCHEMBL10505424 0.84 RAB9A (0.50) RAB9ANPC1SMN1; SMN2OPRD1OPRK1
SCHEMBL28419652 0.84 RAB9A (0.53) RAB9ANPC1SMN1; SMN2
SCHEMBL28418471 0.84 RAB9A (0.49) RAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1083897-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-01-02 EP disclosed
EP-1083897-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-21 EP disclosed
WO-1999062513-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed