SCHEMBL7186786

SCHEMBL7186786

COc1c(C)cc(C)cc1C=CC(=O)c1ccc(C(=O)N(C)C)cc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
ABCG2 Q9UNQ0 3/20 0.48
KRAS P01116 1/20 0.45
CYP1A1 P04798 1/20 0.43
CYP1B1 Q16678 1/20 0.43
CAPN1 P07384 1/20 0.43
GABRA3 P34903 1/20 0.43
GABRA2 P47869 1/20 0.43
GABRB2 P47870 1/20 0.43
TNFRSF1A P19438 1/20 0.43
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ALOX5 P09917 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7185139 0.87 LMNA (0.47) CYP1A1CYP1B1
SCHEMBL7184621 0.87 CYP1A1 (0.41) CA1CA2ABCG2CYP1A1CYP1B1
SCHEMBL7187235 0.85 DPP4 (0.42) ABCG2CYP1A1CYP1B1
SCHEMBL7190651 0.81 ABCG2 (0.61) CA1CA2ABCG2CAPN1TNFRSF1A
SCHEMBL7178660 0.79 ABCG2 (0.66) ABCG2CYP1A1CYP1B1CAPN1TNFRSF1A
SCHEMBL7178662 0.79 ABCG2 (0.66) ABCG2CYP1A1CYP1B1CAPN1TNFRSF1A
SCHEMBL7179752 0.78 ABCG2 (0.60) ABCG2KRASCAPN1TNFRSF1ACTSL
SCHEMBL7179754 0.78 ABCG2 (0.60) ABCG2KRASCAPN1TNFRSF1ACTSL
SCHEMBL7177307 0.77 ABCG2 (0.45) ABCG2KRASCAPN1GABRA3GABRA2
SCHEMBL7190670 0.77 ALDH1A1 (0.43) CA1CA2ABCG2KRASCAPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP disclosed
US-5985935-A PARASITICIDES OR BACTERICIDES STATENS SERUMINSTITUT (DK) 1999-11-16 US disclosed