SCHEMBL7187264

SCHEMBL7187264

O=C(O)CCc1ccc(Oc2c(-c3ccc(F)cc3)ccc3ccccc23)cc1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 16/20 0.56
FFAR4 Q5NUL3 12/20 0.56
AKR1B1 P15121 1/20 0.49
SRD5A2 P31213 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7189113 0.92 FFAR1 (0.57) FFAR1FFAR4AKR1B1SRD5A2
SCHEMBL7190482 0.90 ESR1 (0.53) FFAR1FFAR4AKR1B1SRD5A2
SCHEMBL7188049 0.89 FFAR1 (0.56) FFAR1FFAR4AKR1B1SRD5A2
SCHEMBL7195082 0.86 ESR1 (0.56) FFAR1FFAR4
SCHEMBL7194015 0.85 FFAR1 (0.53) FFAR1FFAR4
SCHEMBL7189203 0.84 ESR1 (0.47) FFAR1FFAR4
SCHEMBL7190740 0.83 FFAR1 (0.53) FFAR1FFAR4AKR1B1
SCHEMBL7183920 0.81 FFAR1 (0.50) FFAR1FFAR4AKR1B1SRD5A2
SCHEMBL6239365 0.80 SRD5A2 (0.49) AKR1B1SRD5A2
SCHEMBL8500438 0.79 MAPT (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0835867-B1 1-Aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods LILLY CO ELI (US) 2003-12-03 EP claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
EP-0835867-A1 1-Aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods ELI LILLY AND COMPANY (US) 1998-04-15 EP claimed
EP-0835867-B1 1-Aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods LILLY CO ELI (US) 2003-12-03 EP disclosed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed
EP-0835867-A1 1-Aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed