SCHEMBL719306

SCHEMBL719306

Cc1cnc(OC2CCC(=O)CC2)nc1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRM7 Q14831 1/20 0.34
PDE10A Q9Y233 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
ACACB O00763 10/20 0.33
MAPK1 P28482 1/20 0.31
HMOX1 P09601 1/20 0.31
CSF1R P07333 1/20 0.31
OGA O60502 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22663349 0.85 CYP11B1 (0.36) GRM7CYP11B1CYP11B2ACACBMAPK1
SCHEMBL631937 0.84 HMOX1 (0.42) PDE4APDE4BPDE4CPDE4DACACB
SCHEMBL720181 0.81 PDE10A (0.37) PDE10APDE4APDE4BPDE4CPDE4D
SCHEMBL17972939 0.81 ACACB (0.41) ACACB
SCHEMBL718781 0.79 EPHX2 (0.38) PDE4APDE4BPDE4CPDE4DHMOX1
SCHEMBL632414 0.78 HCRTR1 (0.42) PDE10A
SCHEMBL718087 0.78 GSK3B (0.36) GRM7CYP11B1CYP11B2ACACBMAPK1
SCHEMBL21192324 0.78 GSK3B (0.36) GRM7CYP11B1CYP11B2ACACBMAPK1
SCHEMBL10052756 0.78 MCHR1 (0.36) GRM7CYP11B1CYP11B2ACACBMAPK1
SCHEMBL29003859 0.76 HRH1 (0.43) CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120053180-A1 CYCLOHEXANE ANALOGUES AS GPR119 AGONISTS CHEMIZON, A DIVISION OF OPTOMAGIC CO., LTD. (KR) 2012-03-01 US disclosed
US-20120053180-A1 CYCLOHEXANE ANALOGUES AS GPR119 AGONISTS CHEMIZON, A DIVISION OF OPTOMAGIC CO., LTD. (KR) 2012-03-01 US disclosed
US-20120053180-A1 CYCLOHEXANE ANALOGUES AS GPR119 AGONISTS CHEMIZON, A DIVISION OF OPTOMAGIC CO., LTD. (KR) 2012-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120053180-A1 CYCLOHEXANE ANALOGUES AS GPR119 AGONISTS GPR119, GLP1R, GIPR GRM7 633/4885PDE10A 772/4885PDE4A 630/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.