SCHEMBL7196637

SCHEMBL7196637

COc1cc(CCC(=O)c2c(OC)ccc(OC)c2OC)c(OC)c(OC)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.54
NPC1 O15118 1/20 0.43
PKM P14618 1/20 0.43
RAB9A P51151 1/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
HSD17B10 Q99714 1/20 0.42
ALOX5 P09917 2/20 0.42
CYP19A1 P11511 1/20 0.42
CYP2D6 P10635 2/20 0.41
LMNA P02545 1/20 0.41
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2C P18825 1/20 0.41
OPRK1 P41145 1/20 0.41
KCNH2 Q12809 1/20 0.41
EBP Q15125 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7195685 0.90 CYP1A2 (0.58) CYP1A2NPC1PKMRAB9ANFKB1
SCHEMBL7193532 0.87 HSD17B10 (0.54) NPC1PKMRAB9AHSD17B10MTNR1A
SCHEMBL7197963 0.82 HSD17B10 (0.54) NPC1PKMRAB9AHSD17B10MTNR1A
SCHEMBL7194480 0.81 CYP1A2 (0.58) CYP1A2NPC1PKMRAB9AHSD17B10
SCHEMBL7190602 0.81 CYP1A2 (0.51) CYP1A2NPC1PKMRAB9AMEN1
SCHEMBL490551 0.81 CYP1A2 (0.61) CYP1A2NPC1PKMRAB9AHSD17B10
SCHEMBL7191887 0.80 NPC1 (0.57) CYP1A2NPC1PKMRAB9A
SCHEMBL7191882 0.78 CYP19A1 (0.46) PKMNFKB1NFKB2RELACYP19A1
SCHEMBL7192539 0.78 CTNNB1 (0.52) CYP1A2NPC1PKMRAB9ALMNA
SCHEMBL7190618 0.77 MTNR1A (0.42) CYP1A2NPC1PKMRAB9AALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030065039-A1 Biologically active 1,3-bis-aromatic-prop-2-en-1-ones, 1,3-bis-aromatic-propan-1-ones, and 1,3-bis-aromatic-prop-2-yn-1-ones STATENS SERUM INSTITUTE (DK) 2003-04-03 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030065039-A1 Biologically active 1,3-bis-aromatic-prop-2-en-1-ones, 1,3-bis-aromatic-propan-1-ones, and 1,3-bis-aromatic-prop-2-yn-1-ones AKR1C3, AKR1C1, AKR1A1 CYP1A2 315/4885NPC1 3105/4885PKM 749/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.