SCHEMBL7196671

SCHEMBL7196671

O=C(O)C(=O)CC(=O)c1cccc(CCc2ccccc2)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC5 P28715 9/20 0.66
FEN1 P39748 9/20 0.66
PTPN1 P18031 4/20 0.65
HAO1 Q9UJM8 3/20 0.53
TDP1 Q9NUW8 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
CYP3A4 P08684 1/20 0.47
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47
ALOX15 P16050 1/20 0.47
CES1 P23141 1/20 0.47
MAPK1 P28482 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NPC1 O15118 1/20 0.46
CASP3 P42574 1/20 0.46
RAB9A P51151 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6940911 0.87 PTPN1 (0.72) ERCC5FEN1PTPN1HAO1TDP1
SCHEMBL6951660 0.84 ERCC5 (0.71) ERCC5FEN1PTPN1HAO1TDP1
Dimethylamine SCHEMBL6946035 0.84 PTPN1 (0.68) ERCC5FEN1PTPN1HAO1
SCHEMBL12182346 0.81 SMN1; SMN2 (0.51) ERCC5FEN1PTPN1MEN1MAPT
SCHEMBL11109822 0.81 NPC1 (0.50) TDP1NPC1CASP3RAB9ASENP8
SCHEMBL6946229 0.80 PTPN1 (0.84) ERCC5FEN1PTPN1SMN1; SMN2RAB9A
SCHEMBL1109671 0.80 ERCC5 (1.00) ERCC5FEN1PTPN1HAO1TDP1
SCHEMBL19090371 0.79 SMN1; SMN2 (0.50) TDP1MAPTHPGDCES1SMN1; SMN2
SCHEMBL6943340 0.79 PTPN1 (0.74) ERCC5FEN1PTPN1HAO1KDM4E
SCHEMBL7665038 0.79 PTPN1 (0.74) ERCC5FEN1PTPN1HAO1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed