SCHEMBL7199489

SCHEMBL7199489

CN1CCCC1Cn1ccc2ccccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 6/20 1.00
CDK4 P11802 4/20 0.50
CCND1 P24385 4/20 0.50
ADRA2A P08913 1/20 0.49
CNR1 P21554 1/20 0.46
CNR2 P34972 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6897355 1.00 HTR6 (1.00) HTR6CDK4CCND1ADRA2ACNR1
SCHEMBL2911126 0.96 HTR6 (0.92) HTR6CDK4CCND1ADRA2ACNR1
SCHEMBL30641113 0.96 HTR6 (0.92) HTR6CDK4CCND1ADRA2ACNR1
Fumaric Acid SCHEMBL8784881 0.89 HTR6 (0.79) HTR6CNR1CNR2
Fumaric Acid SCHEMBL8784884 0.89 HTR6 (0.79) HTR6CNR1CNR2
SCHEMBL8530808 0.87 HTR6 (0.77) HTR6CDK4CCND1ADRA2A
SCHEMBL2267232 0.81 HTR6 (0.67) HTR6
SCHEMBL2261753 0.81 HTR6 (0.67) HTR6
SCHEMBL7253410 0.81 HTR6 (0.67) HTR6
SCHEMBL7253405 0.81 HTR6 (0.67) HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102936240-A Synthetic method of (R)-5-substituted-3-(N-carbobenzoxy pyrrolidine-2-based carbonyl)-1H-benzpyrole ZHEJIANG ACADEMY MEDICAL SCI 2013-02-20 CN disclosed
US-6608079-B1 Activating serotonin-1F receptors, inhibiting neuronal protein extravasation, treating migraine ELI LILLY AND COMPANY 2003-08-19 US disclosed
US-5607951-A SEROTONIN AGONIST FOR NERVOUS SYSTEM DISORDERS, ANALGESICS AND PSYCHOTHERAPEUTICS PFIZER INC (US) 1997-03-04 US disclosed